SCHEMBL27420102

SCHEMBL27420102

Cc1ccc(O)c([N+](=O)[O-])c1C(C)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.47
ALDH1A1 P00352 5/20 0.41
TDP1 Q9NUW8 2/20 0.41
GPR35 Q9HC97 2/20 0.41
PIM1 P11309 1/20 0.39
DYRK1A Q13627 1/20 0.39
PIM3 Q86V86 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
TSHR P16473 5/20 0.38
CYP3A4 P08684 1/20 0.37
CTSB P07858 1/20 0.36
CTSH P09668 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688608 0.81 TSHR (0.46) ALDH1A1TDP1TSHRCYP3A4GAA
SCHEMBL2881308 0.77 ALDH1A1 (0.56) MCL1ALDH1A1TDP1GPR35PIM1
SCHEMBL6858240 0.76 MCL1 (0.49) MCL1ALDH1A1TDP1GPR35PIM1
SCHEMBL6397577 0.73 TRPA1 (0.40) ALDH1A1TDP1TSHRCYP3A4ESR1
SCHEMBL22363065 0.73 MCL1 (0.46) MCL1ALDH1A1TDP1GPR35PIM1
SCHEMBL28136370 0.73 MCL1 (0.46) MCL1ALDH1A1TDP1GPR35PIM1
SCHEMBL4363348 0.72 GPR35 (0.60) MCL1ALDH1A1TDP1GPR35TSHR
SCHEMBL5206322 0.72 ALDH1A1 (0.54) MCL1ALDH1A1TDP1GPR35PIM1
SCHEMBL28740174 0.72 ALDH1A1 (0.54) MCL1ALDH1A1TDP1GPR35PIM1
Acetic Acid SCHEMBL29244387 0.71 ALDH1A1 (0.48) MCL1ALDH1A1TDP1GPR35PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1079397-C 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives endothelin antagonists ABBOTT LAB (US) 2002-02-20 CN disclosed
CN-1265097-A Pyrrolidine carboxylic acid derivatives as endothelin antagonists ABBOTT LAB (US) 2000-08-30 CN disclosed
CN-1215401-A 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives endothelin antagonists ABBOTT LAB (US) 1999-04-28 CN disclosed