Quinoline

Quinoline

SCHEMBL27434751

CCOC=O.c1ccc2ncccc2c1

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.57
GAA P10253 2/20 0.44
PDE10A Q9Y233 1/20 0.40
HTT P42858 3/20 0.39
CYP3A4 P08684 2/20 0.39
ALOX15 P16050 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 1/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
TLR8 Q9NR97 1/20 0.37
KDM4E B2RXH2 2/20 0.36
CASP1 P29466 2/20 0.36
MEN1 O00255 1/20 0.36
CASP7 P55210 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL27574374 0.98 ALDH1A1 (0.55) ALDH1A1GAAPDE10AHTTCYP3A4
Quinoline SCHEMBL27586146 0.87 ALDH1A1 (0.53) ALDH1A1GAAPDE10AHTTCYP3A4
Quinoxaline SCHEMBL27913231 0.86 ALDH1A1 (0.41) ALDH1A1GAASMN1; SMN2NPC1POLB
Quinoline SCHEMBL27788010 0.84 ALDH1A1 (0.50) ALDH1A1GAAPDE10AHTTCYP3A4
Quinoxaline SCHEMBL27907726 0.84 ALDH1A1 (0.41) ALDH1A1GAASMN1; SMN2NPC1POLB
Ethoxycarbonyl Group SCHEMBL27997141 0.83 ALDH1A1 (0.47) ALDH1A1GAAHTTCYP3A4ALOX15
Quinoline SCHEMBL28060746 0.82 ALDH1A1 (0.65) ALDH1A1GAAPDE10AHTTCYP3A4
Quinoline SCHEMBL6808379 0.82 ALDH1A1 (0.65) ALDH1A1GAAPDE10AHTTCYP3A4
Quinoline SCHEMBL1257445 0.80 ALDH1A1 (0.68) ALDH1A1GAAPDE10AHTTCYP3A4
Quinoline SCHEMBL28250556 0.80 ALDH1A1 (0.74) ALDH1A1PDE10AHTTCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115825057-B Application of quinoline carboxylic ester organic heterocyclic small molecule 郑州轻工业大学 2023-08-22 CN claimed
CN-115825057-A Application of quinoline carboxylic ester organic heterocyclic micromolecules 郑州轻工业大学 2023-03-21 CN claimed
CN-1886124-A Method for inhibiting production of remnant lipoproteins JAPAN TOBACCO INC (JP) 2006-12-27 CN claimed
CN-1635911-A Self-emulsifying formulations of cholesteryl ester transfer protein inhibitors PFIZER PROD INC (US) 2005-07-06 CN claimed
CN-119019327-A Acetylation method of quinoline or isoquinoline compounds 常州工程职业技术学院 2024-11-26 CN disclosed
CN-119019327-A Acetylation method of quinoline or isoquinoline compounds 常州工程职业技术学院 2024-11-26 CN disclosed
CN-115825057-B Application of quinoline carboxylic ester organic heterocyclic small molecule 郑州轻工业大学 2023-08-22 CN disclosed
CN-115825057-A Application of quinoline carboxylic ester organic heterocyclic micromolecules 郑州轻工业大学 2023-03-21 CN disclosed
CN-110003121-A A kind of 3,4- dihydroquinazoline derivatives and preparation method thereof, application 郑州大学 2019-07-12 CN disclosed
CN-109762768-A Bacillus B8W22 and its application 浙江工业大学 2019-05-17 CN disclosed
CN-109689639-A Spirolactams as ROCK inhibitor 百时美施贵宝公司 2019-04-26 CN disclosed
CN-108484497-A A kind of synthetic method of 3- amino -7- chloroquinolines 苏州康润医药有限公司 2018-09-04 CN disclosed
CN-1665536-A Use of CETP inhibitors and antihypertensive agents as well as optionally HMG COA reductase inhibitors PFIZER PROD INC (US) 2005-09-07 CN disclosed
CN-1635911-A Self-emulsifying formulations of cholesteryl ester transfer protein inhibitors PFIZER PROD INC (US) 2005-07-06 CN disclosed
CN-1523979-A Pharmaceutical compositions of adsorbates of amorphous drug �Ʒ� 2004-08-25 CN disclosed
CN-1515259-A 4-aminosubstituted-2-substituted-1,2,3,4-tetrahydroquinoline used as CETP inhibitor �������Զ�˹�Ʒ� 2004-07-28 CN disclosed
CN-1128790-C 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents UPJOHN CO (US) 2003-11-26 CN disclosed
CN-1318058-A 4-carboxyamino-2-substituted-1,2,3,4-tetrahydroquinolines as CRTP inhibitors PFIZER PROD INC (US) 2001-10-17 CN disclosed
CN-1318057-A 4-amino substituted-2-substituted-1, 2,3, 4-tetrahydroquinolines as CETP inhibitors PFIZER PROD INC (US) 2001-10-17 CN disclosed
CN-1281439-A 4-hydroxyquinoline-3-carboxamide and hydrazide compounds as antiviral agents UPJOHN CO (US) 2001-01-24 CN disclosed