SCHEMBL2743933

SCHEMBL2743933

CC(C)(CNc1c(N)cnc2ccccc12)NC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
NPC1 O15118 1/20 0.47
GAA P10253 1/20 0.47
RAB9A P51151 1/20 0.47
LATS1 O95835 1/20 0.46
AAK1 Q2M2I8 2/20 0.44
PKM P14618 1/20 0.39
TOP2A P11388 1/20 0.38
TOP2B Q02880 1/20 0.38
SSTR4 P31391 1/20 0.37
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
BCHE P06276 1/20 0.37
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 2/20 0.37
MAP4K4 O95819 1/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
ACACB O00763 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204017 0.87 MEN1 (0.48) MEN1KMT2ANPC1GAARAB9A
SCHEMBL12757192 0.85 MEN1 (0.48) MEN1KMT2ANPC1GAARAB9A
SCHEMBL24604527 0.84 MEN1 (0.46) MEN1KMT2ANPC1GAARAB9A
SCHEMBL4299216 0.84 LATS1 (0.45) MEN1KMT2ANPC1GAARAB9A
SCHEMBL1232910 0.84 BCHE (0.52) MEN1KMT2ANPC1GAARAB9A
SCHEMBL1041911 0.84 MEN1 (0.45) MEN1KMT2ANPC1GAARAB9A
SCHEMBL1034070 0.82 BRD4 (0.47) MEN1KMT2ANPC1GAARAB9A
SCHEMBL29947676 0.82 HDAC1 (0.48) MEN1KMT2ANPC1GAARAB9A
SCHEMBL1232778 0.82 STK17B (0.47) MEN1KMT2ANPC1GAARAB9A
SCHEMBL29475728 0.82 BRD4 (0.47) MEN1KMT2ANPC1GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230248835-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF FIBROTIC DISEASES AND CANCER PURDUE RESEARCH FOUNDATION 2023-08-10 US disclosed
US-20230248835-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF FIBROTIC DISEASES AND CANCER PURDUE RESEARCH FOUNDATION 2023-08-10 US disclosed
WO-2022147576-A1 METHODS FOR ENHANCEMENT OF ENGINEERED CELL THERAPIES IN CANCER TREATMENT PURDUE RESEARCH FOUNDATION (US) 2022-07-07 WO disclosed
WO-2022011043-A2 COMPOUNDS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF FIBROTIC DISEASES AND CANCER PURDUE RESEARCH FOUNDATION (US) 2022-01-13 WO disclosed
US-8846710-B2 Method of preferentially inducing the biosynthesis of interferon 3M INNOVATIVE PROPERTIES COMPANY (US) 2014-09-30 US disclosed
US-8178677-B2 Hydroxyalkyl substituted imidazoquinolines 3M INNOVATIVE PROPERTIES COMPANY (US) 2012-05-15 US disclosed
US-20090029988-A1 Hydroxyalkyl Substituted Imidazoquinolines COLEY PHARMACEUTICAL GROP, INC. (US) 2009-01-29 US disclosed
US-20090030031-A1 Method of Preferentially Inducing the Biosynthesis of Interferon COLEY PHARMACEUTICAL GROUP, INC. (US) 2009-01-29 US disclosed
US-20070287724-A1 Substituted Imidazoquinolines, Imidazopyridines, and Imidazonaphthyridines 3M INNOVATIVE PROPERTIES COMPANY (US) 2007-12-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230248835-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF FIBROTIC DISEASES AND CANCER TLR9, TLR8, TLR7 MEN1 3475/4885KMT2A 1143/4885NPC1 1683/4885
US-20090030031-A1 Method of Preferentially Inducing the Biosynthesis of Interferon IFNG, IFNAR1, EIF2AK2 MEN1 4113/4885KMT2A 2737/4885NPC1 3690/4885
US-20070287724-A1 Substituted Imidazoquinolines, Imidazopyridines, and Imidazonaphthyridines IL2, IFNG, IL4 MEN1 2129/4885KMT2A 4053/4885NPC1 2144/4885
US-20090029988-A1 Hydroxyalkyl Substituted Imidazoquinolines IFNG, IRF3, IFNAR1 MEN1 4492/4885KMT2A 1364/4885NPC1 2391/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.