SCHEMBL27445164

SCHEMBL27445164

CC(=O)Cl.CS(=O)(=O)NC(Cc1ccccc1)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 9/20 0.57
MMP9 P14780 7/20 0.57
ADAMTS4 O75173 1/20 0.57
POLB P06746 2/20 0.54
ADAMTS5 Q9UNA0 1/20 0.54
ALDH1A1 P00352 1/20 0.54
MAPT P10636 1/20 0.54
HTT P42858 1/20 0.54
ITGB3 P05106 3/20 0.53
ITGA2B P08514 2/20 0.53
MMP1 P03956 1/20 0.51
MMP3 P08254 1/20 0.51
MMP7 P09237 1/20 0.51
MMP13 P45452 1/20 0.51
ITGAV P06756 2/20 0.49
PPARG P37231 1/20 0.48
ITGB1 P05556 1/20 0.47
ITGB5 P18084 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL698061 0.94 MMP2 (0.63) MMP2MMP9ADAMTS4POLBADAMTS5
SCHEMBL6436714 0.94 MMP2 (0.63) MMP2MMP9ADAMTS4POLBADAMTS5
SCHEMBL698062 0.94 MMP2 (0.63) MMP2MMP9ADAMTS4POLBADAMTS5
Benzene SCHEMBL28198278 0.94 MMP2 (0.63) MMP2MMP9ADAMTS4POLBADAMTS5
D-Phenylalanine SCHEMBL8609785 0.88 ALPI (0.63) MMP2MMP9ADAMTS4POLBADAMTS5
SCHEMBL11471487 0.88 POLB (0.49) MMP2MMP9ADAMTS4POLBADAMTS5
SCHEMBL16473194 0.86 MMP2 (0.50) MMP2MMP9ADAMTS4POLBALDH1A1
SCHEMBL27695660 0.85 ITGB3 (0.60) MMP2MMP9ADAMTS4POLBADAMTS5
SCHEMBL27677080 0.84 POLB (0.60) MMP2MMP9ADAMTS4POLBADAMTS5
SCHEMBL9012465 0.84 MME (0.60) MMP2MMP9ADAMTS4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1163466-C Substituted oxobutanoic acid derivatives as matrix metalloproteinase inhibitors 2004-08-25 CN disclosed
CN-1139570-C Inhibition of matrix metalloproteases by acetylene contg. compounds 拜尔公司 2004-02-25 CN disclosed
CN-1124255-C Inhibition of matrix metalloproteases by substituted phenethyl compounds BAYER AG (US) 2003-10-15 CN disclosed
CN-1119313-C Inhibition of matrix metalloproteinases by 2- (omega-aroylalkyl) -4-diaryl-4-oxobutanoic acid BAYER AG (US) 2003-08-27 CN disclosed
CN-1100748-C Inhibition of matrix metalloproteinases by 2-substituted-4- (4-substituted phenyl) -4-oxobutanoic acid BAYER AG (US) 2003-02-05 CN disclosed
CN-1234791-A Inhibition of matrix metalloproteases by 2-('omega'-aroylalkyl)-4-biaryl-oxobutyric acids BAYER AG (US) 1999-11-10 CN disclosed
CN-1225620-A Substituted 4-arylbutanoic acid derivatives as matrix metalloproteinase inhibitors BAYER AG (US) 1999-08-11 CN disclosed
CN-1225621-A Inhibition of matrix metalloproteinases by 2-substituted-4- (4-substituted phenyl) -4-oxobutanoic acid BAYER AG (US) 1999-08-11 CN disclosed
CN-1225622-A Substituted oxobutyric acids as matrix metalloprotease inhibitor BAYER AG (US) 1999-08-11 CN disclosed
CN-1225624-A Inhibition of matrix metalloproteases by substituted phenethyl compounds BAYER AG (US) 1999-08-11 CN disclosed
CN-1225623-A Inhibition of matrix metalloproteases by acetylene contg. compounds BAYER AG (US) 1999-08-11 CN disclosed