SCHEMBL27445188

SCHEMBL27445188

C[C@@H](CCc1cccc(N)c1O)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.42
HMGB1 P09429 1/20 0.41
TSHR P16473 1/20 0.40
GABRR1 P24046 2/20 0.39
GPR35 Q9HC97 1/20 0.39
IAPP P10997 4/20 0.38
GABRA1 P14867 2/20 0.37
GABRB2 P47870 2/20 0.37
ESR1 P03372 1/20 0.35
KCNH2 Q12809 1/20 0.35
LTB4R Q15722 3/20 0.35
CYP1A2 P05177 1/20 0.35
APAF1 O14727 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27442998 1.00 MMP2 (0.42) MMP2HMGB1TSHRGABRR1GPR35
Hydrochloric Acid SCHEMBL27537274 0.98 MMP2 (0.41) MMP2HMGB1TSHRGABRR1GPR35
Acetic Acid SCHEMBL27543237 0.97 MMP2 (0.40) MMP2HMGB1TSHRGABRR1GPR35
SCHEMBL27741080 0.85 TSHR (0.46) TSHRGABRR1GPR35LTB4RCYP1A2
SCHEMBL7038034 0.83 MMP2 (0.43) MMP2HMGB1
SCHEMBL27412207 0.77 AKR1B1 (0.50) TSHRGABRR1LTB4RCYP1A2APAF1
SCHEMBL28115918 0.76 MMP2 (0.39) MMP2HMGB1TSHRIAPPGABRA1
SCHEMBL29133246 0.76 LTB4R (0.47) TSHRGABRR1LTB4RAPAF1
SCHEMBL6248978 0.75 MMP2 (0.48) MMP2HMGB1IAPP
SCHEMBL8442321 0.74 ALDH1A1 (0.41) MMP2TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1098838-C Substituted N- (indole-2-carbonyl) -beta-alaninamides and derivatives as antidiabetics PFIZER (US) 2003-01-15 CN disclosed
CN-1140709-A Substituted N- (indole-2-carbonyl) -beta-alaninamides and derivatives as antidiabetics PFIZER (US) 1997-01-22 CN disclosed