SCHEMBL2745007

SCHEMBL2745007

CCCc1cc(-c2ccc[c]n2)c(C2CCC2)cc1OCCN(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.41
HTR1B P28222 2/20 0.41
NOS3 P29474 6/20 0.38
NOS1 P29475 6/20 0.38
NOS2 P35228 4/20 0.36
HTR7 P34969 3/20 0.35
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
DRD4 P21917 1/20 0.34
DRD5 P21918 1/20 0.34
ABCB11 O95342 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
SCN1A P35498 1/20 0.33
SCN2A Q99250 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
SCN3A Q9NY46 1/20 0.33
PPARG P37231 3/20 0.33
PPARD Q03181 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL221165 0.83 NOS1 (0.58) HTR1DHTR1BNOS3NOS1NOS2
SCHEMBL2744102 0.82 NOS1 (0.56) NOS3NOS1NOS2HTR7ABCB11
SCHEMBL27981902 0.81 ABCB11 (0.43) NOS3NOS1NOS2HTR7DRD2
SCHEMBL27981553 0.74 NOS1 (0.67) NOS3NOS1NOS2HTR7DRD2
SCHEMBL27981883 0.70 PTPN1 (0.43) NOS3NOS1NOS2KDM4EALDH1A1
SCHEMBL27981551 0.69 KDM4E (0.43) HTR1BNOS3NOS1NOS2HTR7
SCHEMBL4282781 0.69 NOS1 (0.54) NOS3NOS1NOS2HTR7LMNA
SCHEMBL27981576 0.68 NOS3 (0.44) HTR1BNOS3NOS1NOS2HTR7
SCHEMBL27981549 0.67 PTPN1 (0.41) NOS3NOS1NOS2LMNAKDM4E
SCHEMBL7074878 0.67 NOS1 (0.42) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178536-B2 Sirtuin modulating compounds SIRTRIS PHARMACEUTICALS, INC. (US) 2012-05-15 US disclosed