SCHEMBL27460864

SCHEMBL27460864

CCOP(=O)(COc1ccccc1)c1ccc(CCNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.47
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
MAPT P10636 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
NAMPT P43490 1/20 0.45
CTSK P43235 1/20 0.44
KMT2A Q03164 3/20 0.42
GLA P06280 1/20 0.42
ADAM17 P78536 2/20 0.42
MMP1 P03956 1/20 0.42
MMP3 P08254 1/20 0.42
MMP9 P14780 1/20 0.42
GAA P10253 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
MEN1 O00255 2/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
CA1 P00915 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8230392 0.83 GLA (0.47) PTPN1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL27460415 0.82 ACACB (0.45) PTPN1CTSK
SCHEMBL27460037 0.80 PTPN1 (0.47) PTPN1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL14812122 0.80 CA2 (0.48) MAPTNAMPTCTSKKMT2AGLA
SCHEMBL8728998 0.78 CA2 (0.48) PTPN1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL27741033 0.77 ACACB (0.59) NPC1RAB9AMAPTSMN1; SMN2NAMPT
SCHEMBL27479632 0.77 AOX1 (0.42) SMN1; SMN2TAAR1LTA4HEPHX2
SCHEMBL13886599 0.76 EPHX2 (0.59) PTPN1NPC1RAB9ANAMPTCTSK
SCHEMBL5142116 0.76 GLA (0.49) NPC1RAB9AMAPTSMN1; SMN2NAMPT
SCHEMBL14763270 0.76 CA1 (0.49) NPC1RAB9AMAPTSMN1; SMN2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1159797-A Aryloxy and arylthiopropanolamine derivative suseful as beta 3-adrenoreceptor agonists and antagonists of the beta 1 and beta 2-adrenoreceptors and pharmaceutical composition thereof SMITHKLINE BEECHAM PLC (GB) 1997-09-17 CN disclosed