SCHEMBL27465741

SCHEMBL27465741

C#Cc1ccc(C(C)C(=O)C(C)c2ccc(C#C)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.40
PTGS2 P35354 5/20 0.38
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
PTGS1 P23219 4/20 0.36
LMNA P02545 2/20 0.36
AKR1C3 P42330 2/20 0.36
CXCR1 P25024 2/20 0.36
CXCR2 P25025 2/20 0.36
ESR1 P03372 2/20 0.36
ALB P02768 1/20 0.36
ALOX5 P09917 1/20 0.36
RARB P10826 1/20 0.36
ADRB3 P13945 1/20 0.36
NFKB1 P19838 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL455771 0.84 EPHX1 (0.53) CYP2C9PTGS2CA12CA1CA2
SCHEMBL18997714 0.81 CYP2C9 (0.36) CYP2C9PTGS2CA12CA1CA2
SCHEMBL27514070 0.79 GSK3B (0.46) CA12CA1CA2CA9CA14
SCHEMBL27538543 0.77 PTGS1 (0.40) CYP2C9PTGS2CA12CA1CA2
SCHEMBL461182 0.77 CYP2C9 (0.43) CYP2C9TSHR
SCHEMBL16070587 0.76 NOS3 (0.41) CYP2C9CA12CA1CA2CA4
SCHEMBL16070644 0.76 NOS3 (0.41) CYP2C9CA12CA1CA2CA4
SCHEMBL30846910 0.76 NOS3 (0.41) CYP2C9CA12CA1CA2CA4
SCHEMBL27512331 0.75 CYP2C9 (0.48) CYP2C9PTGS2PTGS1LMNAAKR1C3
SCHEMBL624888 0.75 PYCR1 (0.42) CYP2C9CA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1946670-A Method for producing 1, 3-enynes using copper catalysts UNIV MASSACHUSETTS (US) 2007-04-11 CN disclosed
CN-1136198-C Novel benzyl pyrimidines ��������ҩ�ɷ����޹�˾ 2004-01-28 CN disclosed
CN-1166831-A Novel benzyl pyrimidines HOFFMANN LA ROCHE (CH) 1997-12-03 CN disclosed