SCHEMBL27486162

SCHEMBL27486162

O=C(O)/C=C/C1(c2cccc(-c3ccccc3)c2)C=CC=NC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.34
CAMK2A Q9UQM7 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KMO O15229 1/20 0.31
IP6K1 Q92551 3/20 0.31
IP6K3 Q96PC2 3/20 0.31
IP6K2 Q9UHH9 3/20 0.31
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
BACE1 P56817 1/20 0.30
HTT P42858 2/20 0.30
USP2 O75604 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPK1 P28482 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27484414 0.88 HCAR2 (0.33)
SCHEMBL27502713 0.85 HSD11B1 (0.38) CCR2ALDH1A1KDM4EMAPTBACE1
SCHEMBL27502712 0.85 LPAR1 (0.38) IP6K1IP6K3IP6K2ALDH1A1HTT
SCHEMBL27554955 0.83 CCNC (0.34) SLC6A4SLC6A3KDM4ELMNA
SCHEMBL27502711 0.82 HSD11B1 (0.41) SLC6A2SLC6A4SLC6A3ALDH1A1BACE1
SCHEMBL27529131 0.80 ALDH1A1 (0.48) ALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL27502325 0.79 MEN1 (0.35) SLC6A2SLC6A4SLC6A3ALDH1A1LMNA
SCHEMBL27504121 0.77 HSD11B1 (0.33) ALDH1A1MAPT
SCHEMBL27504464 0.77 HSD11B1 (0.35) ALDH1A1MAPTGAALMNA
SCHEMBL27503047 0.75 CRHBP (0.35) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1196721-A Heteroaryl-substituted acryloylguanidine derivatives and medicinal composition thereof YAMANOUCHI PHARMA CO LTD (JP) 1998-10-21 CN disclosed