SCHEMBL27495178

SCHEMBL27495178

CCSC(=N)Nc1ccc(NCc2ccccc2)c(CN)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.37
HDAC8 Q9BY41 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HTR6 P50406 1/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC3 O15379 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
PPM1D O15297 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27495608 0.85 AOC1 (0.35) IDO1MAPTKDM4EALDH1A1HPGD
SCHEMBL6674456 0.82 IDO1 (0.38) IDO1HDAC8MEN1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL6675350 0.81 IDO1 (0.37) IDO1HDAC8SMN1; SMN2MAPTNPC1
SCHEMBL27493974 0.81 AOC1 (0.33) HDAC8HTTHDAC1HDAC2HDAC3
SCHEMBL27544136 0.80 IDO1 (0.41) IDO1HDAC8MAPTKDM4EHDAC1
SCHEMBL27552471 0.78 HDAC3 (0.33) IDO1HDAC8HTTHDAC1HDAC2
SCHEMBL27479163 0.78 C5AR1 (0.47) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL6674459 0.78 CACNA1C (0.43) IDO1HDAC8HTR6
Hydrochloric Acid SCHEMBL27564406 0.77 HDAC3 (0.32) HDAC8HDAC1HDAC2HDAC3
Hydrochloric Acid SCHEMBL6675354 0.77 CACNA1C (0.42) IDO1HDAC8HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1172473-A Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 1998-02-04 CN claimed
CN-1310169-A Anils with nitric oxide synzyme inhibiting function SHUGAI SEIYAKU K K (JP) 2001-08-29 CN disclosed
CN-1172473-A Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 1998-02-04 CN disclosed