SCHEMBL6674459

SCHEMBL6674459

CCN=C(N)Nc1ccc(NCc2ccccc2)c(CN)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.43
SCN5A Q14524 1/20 0.43
PTGIR P43119 2/20 0.39
SIGMAR1 Q99720 4/20 0.39
C5AR1 P21730 3/20 0.39
IDO1 P14902 1/20 0.38
HTR6 P50406 1/20 0.37
CXCR4 P61073 2/20 0.37
HDAC8 Q9BY41 1/20 0.37
ADRA2A P08913 3/20 0.36
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6675354 0.99 CACNA1C (0.42) CACNA1CSCN5APTGIRSIGMAR1C5AR1
SCHEMBL6675283 0.85 ADRA2A (0.47) CACNA1CSCN5APTGIRSIGMAR1ADRA2A
Hydrochloric Acid SCHEMBL6677488 0.84 ADRA2A (0.49) CACNA1CSCN5APTGIRADRA2A
SCHEMBL6676284 0.81 PTGIR (0.45) CACNA1CSCN5APTGIRSIGMAR1CXCR4
SCHEMBL6676123 0.80 KCNK3 (0.50) CACNA1CSCN5AGRIN2DGRIN3BGRIN1
Hydrochloric Acid SCHEMBL6678108 0.80 PTGIR (0.44) CACNA1CSCN5APTGIRSIGMAR1ADRA2A
SCHEMBL6674456 0.79 IDO1 (0.38) IDO1HTR6HDAC8
SCHEMBL6678178 0.78 C5AR1 (0.60) C5AR1
Hydrochloric Acid SCHEMBL6675350 0.78 IDO1 (0.37) IDO1HTR6HDAC8
SCHEMBL27495178 0.78 IDO1 (0.37) IDO1HTR6HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP claimed