SCHEMBL27544136

SCHEMBL27544136

CCSC(=N)Nc1ccc(NCc2ccccc2)c(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.41
NAMPT P43490 2/20 0.41
HDAC1 Q13547 2/20 0.40
GLS O94925 4/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA7 P43166 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CTSK P43235 1/20 0.37
KDM4A O75164 1/20 0.36
SYK P43405 1/20 0.36
MAPT P10636 3/20 0.36
TDP1 Q9NUW8 3/20 0.36
KDM4E B2RXH2 2/20 0.36
ATM Q13315 1/20 0.36
MAPK1 P28482 1/20 0.36
AURKA O14965 1/20 0.35
RPS6KB1 P23443 1/20 0.35
CTSL P07711 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27564883 0.84 CYP2C9 (0.45) IDO1NAMPTHDAC1GLSSYK
SCHEMBL27577235 0.81 IDO1 (0.43) IDO1NAMPTHDAC1GLSKDM4A
SCHEMBL27564542 0.81 JAK2 (0.39) IDO1NAMPTHDAC1GLSKDM4A
SCHEMBL27495178 0.80 IDO1 (0.37) IDO1HDAC1CA1MAPTKDM4E
SCHEMBL27545134 0.79 HDAC1 (0.44) IDO1NAMPTHDAC1GLSKDM4A
SCHEMBL27564508 0.78 ALDH1A1 (0.44) IDO1NAMPTGLSKDM4AMAPT
SCHEMBL7740424 0.75 MEN1 (0.36) NAMPTGLSSYKMAPTMAPK1
SCHEMBL16486018 0.74 AURKA (0.48) NAMPTHDAC1GLSCA12CA1
SCHEMBL28745798 0.73 HDAC1 (0.48) IDO1NAMPTHDAC1GLS
SCHEMBL17141855 0.73 NAMPT (0.48) NAMPTHDAC1CA12CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1310169-A Anils with nitric oxide synzyme inhibiting function SHUGAI SEIYAKU K K (JP) 2001-08-29 CN disclosed