SCHEMBL27499149

SCHEMBL27499149

CC(C)(C)NC(=O)Oc1cc(Cl)c(I)cc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.38
MAPT P10636 3/20 0.38
NPSR1 Q6W5P4 2/20 0.38
GPR55 Q9Y2T6 2/20 0.38
POLB P06746 1/20 0.38
CCR6 P51684 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
CNR2 P34972 1/20 0.36
ALDH1A1 P00352 3/20 0.36
TBXA2R P21731 4/20 0.36
HSP90AA1 P07900 1/20 0.34
HPGD P15428 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27498855 0.86 MEN1 (0.34) MAPTNPSR1HTTALDH1A1TBXA2R
SCHEMBL27500364 0.85 ALDH1A1 (0.37) LMNAMAPTNPSR1ALDH1A1TBXA2R
SCHEMBL27535554 0.85 NPC1 (0.43) LMNAMAPTNPSR1GPR55POLB
SCHEMBL27566023 0.84 POLB (0.40) LMNAMAPTNPSR1GPR55POLB
SCHEMBL27539107 0.82 LMNA (0.41) LMNAMAPTNPSR1GPR55POLB
SCHEMBL27539426 0.82 HCAR3 (0.37) LMNAMAPTNPSR1HTTALDH1A1
SCHEMBL27484338 0.82 ALDH1A1 (0.35) NPSR1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL27539464 0.80 ALDH1A1 (0.41) LMNAMAPTNPSR1GPR55CYP1A2
SCHEMBL27485133 0.78 TBXA2R (0.45) MAPTNPSR1POLBCYP3A4HTT
SCHEMBL27472206 0.78 LMNA (0.49) LMNAMAPTNPSR1POLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1264825-C Dihydro-benzo [ b ] [1,4] diazepin * -2-one derivatives as mGluR2 antagonists II HOFFMANN LA ROCHE (CH) 2006-07-19 CN disclosed
CN-1195522-C Benzodiazepine derivatives usable as parental metabolic glutamate receptor antagonist HOFFMANN LA ROCHE (CH) 2005-04-06 CN disclosed
CN-1535266-A Dihydro-benzo [b][1,4] diazepin-2-one derivatives as mglur 2 antagonists II - 2004-10-06 CN disclosed
CN-1379765-A Benzodiazepine derivatives usable as parental metabolic glutamate receptor antagonist HOFFMANN LA ROCHE (CH) 2002-11-13 CN disclosed