SCHEMBL27501099

SCHEMBL27501099

Nc1c(Cc2ccccc2C(F)(F)F)csc1-n1cncn1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.42
IDO1 P14902 2/20 0.34
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
ADORA1 P30542 1/20 0.32
EGFR P00533 1/20 0.32
AR P10275 1/20 0.32
KMT2A Q03164 1/20 0.32
YTHDC1 Q96MU7 1/20 0.31
P2RX7 Q99572 1/20 0.31
F2 P00734 1/20 0.31
F10 P00742 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
ATM Q13315 1/20 0.30
LMNA P02545 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27377635 0.72 LTA4H (0.48) LTA4HIDO1EGFRARKDM4E
SCHEMBL9831326 0.66 ALDH1A1 (0.51) KMT2AF2F10KDM4EALDH1A1
SCHEMBL28206568 0.66 CYP19A1 (0.53) IDO1KMT2AP2RX7KDM4EALDH1A1
SCHEMBL23144898 0.63 IDO1 (0.49) LTA4HIDO1EGFRARKMT2A
SCHEMBL27404925 0.60 CYP11B1 (0.45) LTA4HIDO1KMT2AALDH1A1LMNA
SCHEMBL3727774 0.59 ALDH1A1 (0.54) LTA4HIDO1ARALDH1A1ATM
SCHEMBL31061820 0.59 GAA (0.44) KDM4EALDH1A1LMNA
SCHEMBL994006 0.59 GAA (0.44) KDM4EALDH1A1LMNA
SCHEMBL15637377 0.58 IDO1 (0.48) LTA4HIDO1ARP2RX7KDM4E
SCHEMBL3249477 0.58 IDO1 (0.48) LTA4HIDO1ARKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1227560-A Thienopyrimidines MERCK PATENT GMBH (DE) 1999-09-01 CN disclosed