SCHEMBL27536633

SCHEMBL27536633

CC(C(=O)C(C)c1ccc(N2CCOC2=O)nc1)c1ccc(N2CCOC2=O)nc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 12/20 0.43
CCNA2 P20248 3/20 0.42
CDK2 P24941 3/20 0.42
CCNA1 P78396 3/20 0.42
CCNB2 O95067 1/20 0.42
CCNE2 O96020 1/20 0.42
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
CCNB3 Q8WWL7 1/20 0.42
CCR6 P51684 1/20 0.39
MAP4K1 Q92918 1/20 0.39
TYK2 P29597 1/20 0.35
EED O75530 1/20 0.34
SUZ12 Q15022 1/20 0.34
EZH2 Q15910 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27536634 0.82 IDH1 (0.43) IDH1CCNA2CDK2CCNA1CCNB2
SCHEMBL27513024 0.79 CCNA2 (0.56) IDH1CCNA2CDK2CCNA1CCNB2
SCHEMBL27513740 0.77 ALDH1A1 (0.55)
SCHEMBL9964663 0.76 DGAT1 (0.40) IDH1
SCHEMBL2645587 0.76 MAP4K1 (0.39) IDH1MAP4K1TYK2EEDSUZ12
SCHEMBL17229262 0.75 IDH1 (0.39) IDH1EEDSUZ12EZH2
SCHEMBL27514421 0.75 MAPT (0.45)
SCHEMBL14923656 0.74 GRIN2D (0.41) IDH1MAP4K1TYK2EEDSUZ12
SCHEMBL2366061 0.74 RAB9A (0.53) MAP4K1
SCHEMBL13424162 0.73 IDH1 (0.38) IDH1MAP4K1EEDSUZ12EZH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1252070-A 5,7-disubstituted 4-aminopyrido [2,3,-d] pyrimidine compounds and their use as adenosine kinase inhibitors ABBOTT LAB (US) 2000-05-03 CN disclosed