SCHEMBL7740424

SCHEMBL7740424

CCSC(=N)Nc1ccc(-n2cccn2)c(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.36
ALDH1A1 P00352 4/20 0.36
MAPT P10636 4/20 0.36
KMT2A Q03164 4/20 0.36
LMNA P02545 2/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NAMPT P43490 2/20 0.36
SYK P43405 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
CCKBR P32239 1/20 0.35
GLS O94925 1/20 0.35
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
BRD4 O60885 1/20 0.35
CYP17A1 P05093 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740469 0.85 HDAC6 (0.34) NAMPTCCKBRGLSHDAC10HDAC6
SCHEMBL7740422 0.83 SYK (0.40) MEN1ALDH1A1MAPTKMT2ALMNA
SCHEMBL7734198 0.82 TSHR (0.34) MEN1ALDH1A1MAPTKMT2ALMNA
SCHEMBL7740426 0.81 PDK1 (0.40) NAMPTSYKPDK1PDK2PDK3
SCHEMBL7740478 0.81 SYK (0.37) MEN1ALDH1A1MAPTKMT2ALMNA
SCHEMBL7739655 0.80 KMT2A (0.36) MEN1ALDH1A1MAPTKMT2ALMNA
SCHEMBL7740427 0.80 NOS1 (0.38) SYK
SCHEMBL27525664 0.80 RXFP1 (0.35) MEN1ALDH1A1MAPTKMT2ALMNA
SCHEMBL27564542 0.79 JAK2 (0.39) KMT2ANAMPTGLS
SCHEMBL27577235 0.79 IDO1 (0.43) MEN1ALDH1A1KMT2ALMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed