Quinoline

Quinoline

SCHEMBL27550545

c1ccc(-c2cccc3cnccc23)cc1.c1ccc2ncccc2c1

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.58
IKBKE Q14164 1/20 0.51
TBK1 Q9UHD2 1/20 0.51
ALDH1A1 P00352 2/20 0.50
CYP2A6 P11509 1/20 0.44
KDM4E B2RXH2 2/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPKAPK2 P49137 1/20 0.42
NPC1 O15118 1/20 0.42
PIK3CA P42336 2/20 0.42
KCNA3 P22001 1/20 0.42
TOP1 P11387 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL28340669 0.88 TNF (0.77) TNFIKBKETBK1ALDH1A1CYP2A6
SCHEMBL6998015 0.87 TNF (0.73) TNFIKBKETBK1ALDH1A1KDM4E
Quinoline SCHEMBL27278136 0.85 PRKCZ (0.55) TNFIKBKETBK1ALDH1A1CYP2A6
SCHEMBL12074747 0.84 TNF (0.69) TNFIKBKETBK1ALDH1A1KDM4E
SCHEMBL27920029 0.81 PDGFRB (0.59) TNFIKBKETBK1CYP2A6KDM4E
Quinoline SCHEMBL28895783 0.81 ALDH1A1 (0.71) TNFALDH1A1CYP2A6KDM4ELMNA
SCHEMBL17945511 0.80 TNF (0.63) TNFIKBKETBK1ALDH1A1KDM4E
SCHEMBL15835309 0.79 KDM4E (0.56) TNFIKBKETBK1ALDH1A1CYP2A6
Quinoline SCHEMBL28089647 0.79 CYP3A4 (0.54) TNFALDH1A1KDM4ELMNACYP3A4
SCHEMBL17944989 0.79 NPC1 (0.46) TNFIKBKETBK1ALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108017479-A The manufacture method of aromatic compound 东曹株式会社 2018-05-11 CN disclosed
CN-1275979-A Isoquinoline compounds useful as urokinase inhibitors PFIZER (US) 2000-12-06 CN disclosed