Quinoline

Quinoline

SCHEMBL28340669

c1ccc(-c2cccc3ccncc23)cc1.c1ccc2ncccc2c1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 3/20 0.77
ALDH1A1 P00352 2/20 0.50
MAPK10 P53779 1/20 0.47
CYP2A6 P11509 1/20 0.44
NPC1 O15118 1/20 0.42
PIK3CA P42336 2/20 0.42
TOP1 P11387 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP3A4 P08684 1/20 0.40
KCNA5 P22460 1/20 0.40
KCNH2 Q12809 1/20 0.40
HASPIN Q8TF76 1/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL27550545 0.88 TNF (0.58) TNFALDH1A1CYP2A6NPC1PIK3CA
SCHEMBL14740148 0.87 TNF (1.00) TNFALDH1A1MAPK10NPC1KDM4E
SCHEMBL30933417 0.87 TNF (1.00) TNFALDH1A1MAPK10NPC1KDM4E
Quinoline SCHEMBL28089647 0.82 CYP3A4 (0.54) TNFALDH1A1NPC1TOP1KDM4E
Quinoline SCHEMBL28895783 0.81 ALDH1A1 (0.71) TNFALDH1A1CYP2A6NPC1TOP1
Quinoline SCHEMBL29173271 0.80 CYP3A4 (0.59) TNFALDH1A1MAPK10CYP2A6NPC1
SCHEMBL15835315 0.79 TNF (0.77) TNFALDH1A1CYP2A6KDM4EMAPT
SCHEMBL27976477 0.79 TNF (0.82) TNFALDH1A1MAPK10NPC1PIK3CA
SCHEMBL16483488 0.78 TNF (0.52) TNFMAPK10PIK3CACYP3A4CA12
SCHEMBL16483498 0.77 TNF (0.51) TNFMAPK10CYP2A6NPC1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110475773-A 8- phenyl isoquinolin quinoline and its medical composition are for treating irritable bowel syndrome YU LINDA CHIA HUI 2019-11-19 CN disclosed
CN-110475773-A 8- phenyl isoquinolin quinoline and its medical composition are for treating irritable bowel syndrome YU LINDA CHIA HUI 2019-11-19 CN disclosed