SCHEMBL27552138

SCHEMBL27552138

COc1nc2ccccc2c(C)c1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.60
ALDH1A1 P00352 2/20 0.45
CYP1A2 P05177 2/20 0.45
ADORA3 P0DMS8 1/20 0.45
CYP2C19 P33261 1/20 0.45
MAPT P10636 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
MAPK1 P28482 2/20 0.45
KDM4E B2RXH2 1/20 0.45
RAD52 P43351 1/20 0.43
GPR3 P46089 1/20 0.42
LMNA P02545 4/20 0.42
HTT P42858 1/20 0.42
NR1I3 Q14994 2/20 0.42
CYP3A4 P08684 1/20 0.42
VDR P11473 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2B6 P20813 1/20 0.42
AHR P35869 1/20 0.42
SQOR Q9Y6N5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4272933 0.85 POLB (0.66) POLBALDH1A1CYP1A2ADORA3CYP2C19
SCHEMBL29450270 0.85 POLB (0.70) POLBALDH1A1CYP1A2ADORA3CYP2C19
SCHEMBL9694998 0.85 POLB (0.70) POLBALDH1A1CYP1A2ADORA3CYP2C19
SCHEMBL21940616 0.83 POLB (0.62) POLBALDH1A1CYP1A2MAPTSMN1; SMN2
SCHEMBL29693599 0.80 POLB (0.58) POLBALDH1A1CYP1A2ADORA3CYP2C19
SCHEMBL8136134 0.77 ALDH1A1 (0.55) POLBALDH1A1CYP1A2ADORA3CYP2C19
SCHEMBL23145043 0.76 POLB (0.63) POLBALDH1A1CYP1A2ADORA3CYP2C19
SCHEMBL7048658 0.76 CYP1A2 (0.58) POLBALDH1A1CYP1A2ADORA3CYP2C19
SCHEMBL9762619 0.76 POLB (0.53) POLBALDH1A1CYP1A2ADORA3CYP2C19
SCHEMBL22377 0.76 PDE10A (0.57) POLBALDH1A1SMN1; SMN2KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1176922-C 8-quinolinxanthine and 8-isoquinolinxanthine derivs. as PDE 5 inhibitors ��˹��ŵ�� 2004-11-24 CN disclosed
CN-1420887-A 8-quinolinxanthine and 8-isoquinolinxanthine derivs. as PDE 5 inhibitors NOVARTIS AG (CH) 2003-05-28 CN disclosed