SCHEMBL8136134

SCHEMBL8136134

COc1nc2ccccc2c(C)c1C#N

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
KDM4E B2RXH2 2/20 0.55
SQOR Q9Y6N5 7/20 0.53
RECQL P46063 1/20 0.46
POLB P06746 1/20 0.46
ADORA3 P0DMS8 1/20 0.42
MAPT P10636 2/20 0.42
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7830291 0.83 POLB (0.59) ALDH1A1KDM4ESQORRECQLPOLB
SCHEMBL9029678 0.82 KDM4E (0.53) ALDH1A1KDM4ESQORRECQLPOLB
SCHEMBL3970610 0.81 ALDH1A1 (0.60) ALDH1A1KDM4EMAPTCYP1A2CYP2C19
SCHEMBL8129316 0.80 KDM4E (0.56) KDM4ESQORRECQLPOLBMAPT
SCHEMBL6253855 0.78 KDM4E (0.56) ALDH1A1KDM4EPOLBMAPTCYP1A2
SCHEMBL2639136 0.78 ALDH1A1 (0.56) ALDH1A1KDM4ESQORMAPTCYP1A2
SCHEMBL4744765 0.78 ALDH1A1 (0.56) ALDH1A1KDM4EPOLBMAPTCYP1A2
SCHEMBL30315435 0.78 KDM4E (0.56) ALDH1A1KDM4EPOLBMAPTCYP1A2
SCHEMBL7915032 0.78 ALDH1A1 (0.56) ALDH1A1KDM4EMAPTCYP1A2GAA
SCHEMBL27552138 0.77 POLB (0.60) ALDH1A1KDM4ESQORPOLBADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760819-B1 TRICYCLIC DICARBONYL DERIVATIVES HOFFMANN LA ROCHE (CH) 2000-07-19 EP disclosed
US-5688803-A BRAIN DISORDERS; PSYCHOLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 1997-11-18 US disclosed
EP-0760819-A1 TRICYCLIC DICARBONYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed
WO-1995032205-A1 TRICYCLIC DICARBONYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1995-11-30 WO disclosed