SCHEMBL27554657

SCHEMBL27554657

S=C(Nc1ccccc1)Nn1ccnc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.66
ALDH1A1 P00352 6/20 0.66
HPGD P15428 1/20 0.66
QPCT Q16769 1/20 0.53
CYP3A4 P08684 1/20 0.50
TAS2R38 P59533 1/20 0.50
HSD17B10 Q99714 1/20 0.50
GAA P10253 5/20 0.47
KMT2A Q03164 4/20 0.47
MAOA P21397 2/20 0.47
MAOB P27338 2/20 0.47
LMNA P02545 1/20 0.47
MEN1 O00255 3/20 0.47
RAB9A P51151 2/20 0.47
NOX1 Q9Y5S8 2/20 0.47
NPC1 O15118 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.45
CA9 Q16790 1/20 0.45
PTPN7 P35236 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28644193 0.81 TAAR1 (0.54) MAPTCYP3A4KMT2AMAOAMAOB
SCHEMBL28033893 0.80 ALDH1A1 (1.00) MAPTALDH1A1HPGDCYP3A4TAS2R38
SCHEMBL2404117 0.73 CYP3A4 (0.45) MAPTALDH1A1QPCTCYP3A4HSD17B10
SCHEMBL28704185 0.73
SCHEMBL8956322 0.72 ALDH1A1 (0.94) MAPTALDH1A1CYP3A4TAS2R38HSD17B10
SCHEMBL16566469 0.71 ALDH1A1 (0.74) MAPTALDH1A1CYP3A4TAS2R38HSD17B10
SCHEMBL27482733 0.70 CYP26A1 (0.42) MAPTALDH1A1QPCTCYP3A4HSD17B10
SCHEMBL6598806 0.70 TSHR (0.53) MAPTALDH1A1CYP3A4HSD17B10KMT2A
SCHEMBL76301 0.70 QPCT (1.00) ALDH1A1QPCTGAAKMT2AMAOA
SCHEMBL21641770 0.70 HKDC1 (0.42) MAPTQPCTCYP3A4LMNACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1332952-C 4-substituted imidazole-2-thiones, 4-substituted imidazole-2-ones and related compounds and their use ALLERGAN INC (US) 2007-08-22 CN disclosed
CN-1671671-A 4- (substituted cycloalkylmethyl) imidazole-2-thiones, 4- (substituted cycloalkenylmethyl) imidazole-2-thiones, 4- (substituted cycloalkylmethyl) imidazol-2-ones, and 4- (substituted cycloalkenylmethyl) imidazol-2-ones, and related compounds ALLERGAN INC (US) 2005-09-21 CN disclosed