SCHEMBL16566469

SCHEMBL16566469

S=C(Nc1ccccc1)Nc1ccncc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.74
CYP3A4 P08684 2/20 0.74
HSD17B10 Q99714 2/20 0.74
TAS2R38 P59533 1/20 0.74
CA9 Q16790 2/20 0.66
TAAR1 Q96RJ0 1/20 0.64
EPHX1 P07099 2/20 0.64
GAA P10253 5/20 0.62
CA1 P00915 1/20 0.62
KMT2A Q03164 5/20 0.61
MEN1 O00255 3/20 0.61
RAB9A P51151 3/20 0.61
NPC1 O15118 2/20 0.61
NOX1 Q9Y5S8 1/20 0.61
MAOA P21397 2/20 0.61
MAOB P27338 2/20 0.61
LMNA P02545 2/20 0.61
MAPT P10636 2/20 0.59
HTT P42858 2/20 0.56
CYP1A2 P05177 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL132620 0.86 ALDH1A1 (1.00) ALDH1A1CYP3A4HSD17B10TAS2R38GAA
SCHEMBL8956322 0.84 ALDH1A1 (0.94) ALDH1A1CYP3A4HSD17B10TAS2R38GAA
SCHEMBL9470190 0.84 ALDH1A1 (0.94) ALDH1A1CYP3A4HSD17B10TAS2R38GAA
SCHEMBL11186307 0.82 PKM (0.69) ALDH1A1CYP3A4HSD17B10TAS2R38KMT2A
SCHEMBL11095557 0.80 ALDH1A1 (0.63) ALDH1A1CYP3A4HSD17B10TAS2R38GAA
SCHEMBL6297654 0.80 CA9 (1.00) ALDH1A1CA9GAAKMT2AMEN1
Thiourea SCHEMBL21055683 0.79 ALDH1A1 (0.85) ALDH1A1CYP3A4HSD17B10TAS2R38GAA
SCHEMBL9297614 0.79 MDM2 (0.56) ALDH1A1CA9TAAR1EPHX1GAA
SCHEMBL6815965 0.79 MAPT (0.66) ALDH1A1CYP3A4HSD17B10TAS2R38CA9
SCHEMBL29924720 0.79 SMN1; SMN2 (0.62) ALDH1A1CYP3A4HSD17B10TAS2R38CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150080580-A1 THIOUREA DERIVATIVES AS a-CHYMOTRYPSIN INHIBITORS RAHMAN ATTA-UR (PK) 2015-03-19 US disclosed
US-20150080580-A1 THIOUREA DERIVATIVES AS a-CHYMOTRYPSIN INHIBITORS RAHMAN ATTA-UR (PK) 2015-03-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150080580-A1 THIOUREA DERIVATIVES AS a-CHYMOTRYPSIN INHIBITORS SERPINB1, CTRL, RNASE1 ALDH1A1 1629/4885CYP3A4 154/4885HSD17B10 3431/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.