SCHEMBL27559486

SCHEMBL27559486

Cc1c(N=C=O)n(N(C)C)c2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 1/20 0.35
GPR3 P46089 1/20 0.34
TSPO P30536 2/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.31
ALKBH5 Q6P6C2 1/20 0.31
FTO Q9C0B1 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
DNM1 Q05193 2/20 0.30
CHRM2 P08172 1/20 0.30
CHRNA7 P36544 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19154998 0.72 GPR3 (0.55) CYP3A4KDM4EALDH1A1GPR3TSPO
SCHEMBL6008133 0.67 GPR3 (0.44) KDM4EALDH1A1GPR3TSPOPOLB
SCHEMBL9824751 0.65 CYP3A4 (0.50) CYP3A4ALDH1A1TSHRMAPTL3MBTL1
SCHEMBL27559456 0.64 KMT2A (0.44) KDM4EALDH1A1TSPOPOLBTSHR
SCHEMBL28858948 0.61 KDM4E (0.53) CYP3A4KDM4EALDH1A1GPR3POLB
SCHEMBL9731262 0.61 IMPDH2 (0.47) CYP3A4KDM4EALDH1A1POLBLMNA
SCHEMBL11118968 0.61 CYP3A4 (0.45) CYP3A4TSHRL3MBTL1
SCHEMBL17473057 0.61 CYP3A4 (0.45) CYP3A4TSHRL3MBTL1
Hexamethylbenzene SCHEMBL28101399 0.60 CYP3A4 (0.74) CYP3A4ALDH1A1POLBTSHR
SCHEMBL17473106 0.60 CYP1A2 (0.40) CYP3A4KDM4EALDH1A1POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1204121-C 1,4-substituted cyclic amine derivatives EISAI CO LTD (JP) 2005-06-01 CN disclosed
CN-1253547-A 1,4-substituted cyclic amine derivatives EISAI CO LTD (JP) 2000-05-17 CN disclosed