SCHEMBL27563239

SCHEMBL27563239

NC(=O)c1cccc2c1c1[c]cccc1n2Cc1c(F)cc(F)cc1F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.33
ABCC1 P33527 1/20 0.33
CA5A P35218 1/20 0.32
SCN9A Q15858 1/20 0.32
PARP1 P09874 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
XBP1 P17861 1/20 0.31
KMT2A Q03164 1/20 0.31
PLA2G2A P14555 4/20 0.31
MAPK8 P45983 1/20 0.31
PDE4A P27815 1/20 0.30
PDE7A Q13946 1/20 0.30
MAPK14 Q16539 1/20 0.30
DGAT1 O75907 1/20 0.30
GPR52 Q9Y2T5 1/20 0.30
AURKA O14965 1/20 0.30
RPS6KB1 P23443 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2590504 0.92 CA5A (0.38) CYP3A4ABCC1CA5AOPRM1OPRD1
SCHEMBL27530595 0.89 GPR52 (0.37) CYP3A4ABCC1SCN9APARP1LMNA
SCHEMBL27505187 0.88 MAPK14 (0.33) CYP3A4ABCC1SCN9AMAPK14GPR52
SCHEMBL27525922 0.88 AKR1B10 (0.32) CYP3A4ABCC1CA5ASCN9APARP1
SCHEMBL27530519 0.87 SCN9A (0.33) CYP3A4ABCC1SCN9APARP1MEN1
SCHEMBL27506428 0.87 AURKA (0.41) CYP3A4ABCC1SCN9APARP1MAPK8
SCHEMBL27505648 0.87 ABCC1 (0.36) CYP3A4ABCC1CA5ASCN9APARP1
SCHEMBL27505972 0.87 CYP3A4 (0.33) CYP3A4ABCC1CA5AMEN1LMNA
SCHEMBL28740750 0.86 KMT2A (0.34) CYP3A4ABCC1MEN1LMNAXBP1
SCHEMBL28740784 0.86 PDE4A (0.32) CYP3A4ABCC1CA5ASCN9APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1240210-A Substituted tricyclic compound LILLY CO ELI (US) 2000-01-05 CN disclosed