SCHEMBL27569167

SCHEMBL27569167

CC(=O)Nc1ccc(-c2c(C#N)c(N)nc([SH]3C=CC=C3)c2C#N)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.59
ADORA2A P29274 1/20 0.59
ADORA2B P29275 1/20 0.59
ELAVL1 Q15717 1/20 0.46
ADORA1 P30542 2/20 0.44
ALDH1A1 P00352 7/20 0.43
PDE5A O76074 1/20 0.42
PDE1A P54750 1/20 0.42
PDE1B Q01064 1/20 0.42
PDE1C Q14123 1/20 0.42
GHSR Q92847 1/20 0.40
KDM4E B2RXH2 6/20 0.39
MAPT P10636 6/20 0.39
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
HSD17B10 Q99714 4/20 0.39
HPGD P15428 4/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
NPSR1 Q6W5P4 3/20 0.39
RXFP1 Q9HBX9 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013023 0.81 ADORA3 (0.65) ADORA3ADORA2AADORA2BELAVL1ADORA1
SCHEMBL28185528 0.81 ADORA1 (0.52) ADORA3ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4306407 0.80 ADORA3 (0.64) ADORA3ADORA2AADORA2BELAVL1ADORA1
SCHEMBL28325319 0.80 KDM4E (0.56) ADORA2AELAVL1ADORA1ALDH1A1KDM4E
SCHEMBL28185532 0.79 KDM4E (0.55) ADORA3ADORA2AADORA2BELAVL1ADORA1
SCHEMBL28184877 0.78 ADORA2A (0.54) ADORA2AADORA1ALDH1A1KDM4EMEN1
SCHEMBL28184873 0.78 KDM4E (0.54) ADORA2AADORA1ALDH1A1KDM4EMAPT
SCHEMBL13914391 0.76 ADORA2B (0.73) ADORA3ADORA2AADORA2BELAVL1ADORA1
SCHEMBL3556602 0.74 ADORA2B (0.68) ADORA3ADORA2AADORA2BELAVL1ADORA1
SCHEMBL13914390 0.74 ADORA2B (0.77) ADORA3ADORA2AADORA2BELAVL1ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1407971-A Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof BAYER AG (DE) 2003-04-02 CN disclosed