SCHEMBL27587770

SCHEMBL27587770

CC(O)(CC(F)(F)F)C(=O)Nc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 8/20 0.63
PDK2 Q15119 8/20 0.63
PDK3 Q15120 8/20 0.63
PDK4 Q16654 8/20 0.63
ABCC9 O60706 3/20 0.50
ABCC8 Q09428 3/20 0.50
KCNJ11 Q14654 3/20 0.50
KCNJ8 Q15842 3/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
ABCB11 O95342 1/20 0.50
CYP3A4 P08684 3/20 0.49
CYP2C19 P33261 3/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP2C9 P11712 1/20 0.49
HPGD P15428 1/20 0.49
MEN1 O00255 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
TSHR P16473 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322930 0.85 PDK1 (0.60) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL14086870 0.83 PDK1 (0.62) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL14086869 0.83 PDK1 (0.62) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL11874543 0.82 PDK1 (0.57) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL12591123 0.81 PDK1 (0.59) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL18171744 0.80 AR (0.54) PDK1PDK2PDK3PDK4HDAC1
SCHEMBL8575413 0.80 PDK1 (0.54) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL14086879 0.79 PDK1 (0.57) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL14273995 0.79 PDK1 (0.57) PDK1PDK2PDK3PDK4L3MBTL1
SCHEMBL14086866 0.79 PDK1 (0.57) PDK1PDK2PDK3PDK4ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115701991-A Pyrazolylpropionamide compounds and their use for treating prostate cancer 田纳西大学研究基金会 2023-02-14 CN disclosed
CN-101891663-A Preparation method of bicalutamide intermediate Hangzhou minsheng pharmaceutical group co ltd 2010-11-24 CN disclosed
CN-1413188-A Resolution of intermediates in synthesis of substantially pure bicalutamide NOBEX CORP (US) 2003-04-23 CN disclosed
CN-1409702-A Methods for asymmetrically synthesizing enantiomer of casodex, its derivatives and intermediate thereof NOBEX CORP (US) 2003-04-09 CN disclosed