SCHEMBL27597136

SCHEMBL27597136

Cc1ncccc1-c1cccc(C(=O)CC(=O)Nc2cc(Cl)ccc2NC(=O)O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.47
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
ALDH1A1 P00352 1/20 0.47
SERPINE1 P05121 3/20 0.44
RXFP1 Q9HBX9 1/20 0.42
MAPT P10636 3/20 0.41
PTGER1 P34995 2/20 0.41
SUCNR1 Q9BXA5 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
TP53 P04637 1/20 0.39
THRB P10828 1/20 0.39
GRM5 P41594 1/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27615861 0.89 RAB9A (0.42) SMN1; SMN2RAB9ANPC1ALDH1A1RXFP1
SCHEMBL5562371 0.88 SERPINE1 (0.40) SMN1; SMN2RAB9ANPC1ALDH1A1SERPINE1
SCHEMBL27597139 0.86 ALDH1A1 (0.48) SMN1; SMN2RAB9ANPC1ALDH1A1SCN5A
SCHEMBL27615911 0.85 WNT3A (0.44) SMN1; SMN2RAB9ANPC1ALDH1A1SERPINE1
SCHEMBL27615863 0.84 RAB9A (0.46) SMN1; SMN2RAB9ANPC1ALDH1A1SERPINE1
SCHEMBL27597149 0.83 SERPINE1 (0.43) SMN1; SMN2RAB9ANPC1ALDH1A1SERPINE1
SCHEMBL27597111 0.82 SCN5A (0.50) SMN1; SMN2RAB9ANPC1ALDH1A1SCN5A
SCHEMBL27615831 0.82 SCN5A (0.41) SMN1; SMN2RAB9ANPC1ALDH1A1SCN5A
SCHEMBL27597178 0.81 MKNK1 (0.49) PTGER1SCN5ASCN9A
SCHEMBL27615839 0.79 SCN5A (0.47) SMN1; SMN2RAB9ANPC1ALDH1A1SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100497333-C Dihydrobenzodiazepin-2-one derivatives for the treatment of neurological disorders HOFFMANN LA ROCHE (CH) 2009-06-10 CN disclosed
CN-1633430-A Dihydrobenzodiazepin-2-one derivatives for the treatment of neurological disorders HOFFMANN LA ROCHE (CH) 2005-06-29 CN disclosed