SCHEMBL27600173

SCHEMBL27600173

CCn1c(=O)[nH]c(=O)c2c1ncn2CCc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.70
KDM4E B2RXH2 1/20 0.67
LMNA P02545 1/20 0.67
POLB P06746 1/20 0.67
MAPK1 P28482 1/20 0.67
CNOT7 Q9UIV1 7/20 0.64
MEN1 O00255 2/20 0.64
KMT2A Q03164 2/20 0.64
PDE4A P27815 3/20 0.62
ADORA2A P29274 3/20 0.62
PDE4B Q07343 3/20 0.62
PDE4C Q08493 3/20 0.62
PDE4D Q08499 3/20 0.62
ALDH1A1 P00352 2/20 0.60
BRD2 P25440 2/20 0.58
BRD3 Q15059 2/20 0.58
BRDT Q58F21 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27600284 0.87 ALDH1A1 (0.70) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL27256844 0.87 MAPK1 (0.86) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL554932 0.87 BRD4 (0.81) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL27582971 0.86 KDM4E (0.62) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL27600302 0.84 KDM4E (0.60) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL7464482 0.84 PDE4A (0.86) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL27600221 0.83 KDM4E (0.58) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL27583058 0.83 KDM4E (0.58) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL28749938 0.83 LMNA (0.64) BRD4KDM4ELMNAPOLBMAPK1
SCHEMBL516463 0.82 PDE4A (0.81) BRD4MEN1KMT2APDE4AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101293888-B Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA 2013-09-25 CN disclosed
CN-101293888-A Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA (DE) 2008-10-29 CN disclosed
CN-100408579-C Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA (DE) 2008-08-06 CN disclosed
CN-1492870-A Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-04-28 CN disclosed