SCHEMBL27600698

SCHEMBL27600698

CC(C(=O)C(C)c1ccccc1Br)c1ccccc1Br

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.50
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 1/20 0.43
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP26A1 O43174 1/20 0.38
GABRA1 P14867 1/20 0.37
GABRB2 P47870 1/20 0.37
OPRL1 P41146 1/20 0.37
HSD11B1 P28845 2/20 0.36
LMNA P02545 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
PTGS2 P35354 1/20 0.35
F2R P25116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL214223 0.85 HTT (0.49) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL15695565 0.85 HTT (0.49) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL29144510 0.85 HTT (0.49) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL4824347 0.85 HTT (0.49) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL4825414 0.85 HTT (0.49) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL9780867 0.83 HTT (0.51) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL9780871 0.83 HTT (0.51) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL4685959 0.83 HTT (0.47) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL4685960 0.83 CXCL8 (0.47) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL31741597 0.82 GABRA1 (0.43) HTTCYP2C19CYP2C9CYP3A4CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101679395-B Triazolyl aminopyrimidine compounds LILLY CO ELI 2012-06-13 CN disclosed
CN-102498111-A Sulfonamides as inhibitors of Bcl-2 family proteins for the treatment of cancer NOVARTIS AG 2012-06-13 CN disclosed
CN-101679395-A triazolyl aminopyrimidine compounds LILLY CO ELI 2010-03-24 CN disclosed
CN-101208342-A Pyrrolobenzodiazepine * pyridine carboxamides and derivatives as follicle stimulating hormone receptor antagonists WYETH CORP (US) 2008-06-25 CN disclosed
CN-1639146-A Fused tricyclic heterocycles useful for the treatment of hyperproliferative diseases BAYER PHARMACEUTICALS CORP (US) 2005-07-13 CN disclosed