SCHEMBL2760652

SCHEMBL2760652

Cc1ccc([C@H](O)CC(N)=O)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.44
ADRA2A P08913 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
P2RX7 Q99572 3/20 0.38
GRM2 Q14416 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CYP2C19 P33261 1/20 0.37
LGMN Q99538 1/20 0.36
NR3C2 P08235 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10349460 0.85 TSHR (0.42) L3MBTL1P2RX7HDAC1HDAC6KDM4E
SCHEMBL12836123 0.83 P2RX7 (0.40) ADRA2AADRA2BADRA2CP2RX7GRM2
SCHEMBL10349464 0.81 MAPT (0.40) P2RX7HDAC1HDAC6KDM4ESMN1; SMN2
SCHEMBL6075377 0.80 TAAR1 (0.50) L3MBTL1ADRA2AADRA2BADRA2CP2RX7
SCHEMBL2760706 0.80 NNMT (0.51) L3MBTL1KDM4ESMN1; SMN2HTTLMNA
SCHEMBL4531132 0.80 CYP2C19 (0.48) P2RX7CYP2C19SMN1; SMN2HTTLMNA
SCHEMBL10349461 0.80 KDM4E (0.42) P2RX7HDAC1HDAC6CYP2C19KDM4E
SCHEMBL17664582 0.77 CYP3A4 (0.40) ADRA2AADRA2BADRA2CP2RX7GRM2
SCHEMBL1495530 0.77 CYP3A4 (0.40) ADRA2AADRA2BADRA2CP2RX7GRM2
SCHEMBL12352043 0.77 LMNA (0.47) ADRA2AADRA2BADRA2CP2RX7HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262766-A2 AMIDE COMPOUNDS, COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2010-12-22 EP disclosed
WO-2009110985-A2 AMIDE COMPOUNDS, COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2009-09-11 WO disclosed