SCHEMBL27607641

SCHEMBL27607641

COc1ccc(CN2C(O)CN(Cc3ccc(C(=O)O)s3)S2(O)O)c(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
POLB P06746 3/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 2/20 0.38
MAPK1 P28482 1/20 0.38
EPHX2 P34913 2/20 0.38
GAA P10253 1/20 0.38
PTGER4 P35408 1/20 0.38
PTGER2 P43116 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27626464 0.86 ADRA1D (0.38) KMT2AMEN1POLBALDH1A1KDM4E
SCHEMBL27626279 0.82 KMT2A (0.48) KMT2AMEN1POLBALDH1A1KDM4E
SCHEMBL1732588 0.77 EPHX2 (0.44) KMT2AMEN1POLBALDH1A1KDM4E
SCHEMBL27607663 0.74 KMT2A (0.41) KMT2AMEN1POLBALDH1A1KDM4E
SCHEMBL27626544 0.72 KMT2A (0.40) KMT2AMEN1POLBALDH1A1KDM4E
SCHEMBL27626511 0.71 EPHX2 (0.38) KMT2AMEN1POLBALDH1A1KDM4E
SCHEMBL27607658 0.71 KMT2A (0.39) KMT2AMEN1POLBALDH1A1KDM4E
Hydrochloric Acid SCHEMBL27626547 0.67 KMT2A (0.44) KMT2AMEN1POLBALDH1A1KDM4E
SCHEMBL1730991 0.67 EPHX2 (0.42) KMT2AMEN1POLBALDH1A1KDM4E
SCHEMBL21577487 0.64 ALDH1A1 (0.50) KMT2AMEN1POLBALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1646508-A 5-substituted 1, 1-dioxo-1, 2, 5-thiadiazolidin-3-one derivatives as PTP-1B inhibitors NOVARTIS AG (CH) 2005-07-27 CN disclosed