SCHEMBL2760883

SCHEMBL2760883

Cc1ccc(-c2cc(C(=O)NCCc3ccc(C)nc3)cc(C(O)c3ccccc3)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MAPT P10636 3/20 0.45
TP53 P04637 2/20 0.45
AKR1C3 P42330 4/20 0.42
AKR1C4 P17516 3/20 0.42
AKR1C2 P52895 2/20 0.42
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
P2RX3 P56373 1/20 0.41
P2RX2 Q9UBL9 1/20 0.41
EP300 Q09472 1/20 0.41
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2760882 1.00 NPC1 (0.46) NPC1RAB9AMAPTTP53AKR1C3
SCHEMBL12757626 0.90 AKR1C3 (0.50) AKR1C3AKR1C4AKR1C2P2RX3P2RX2
SCHEMBL2760639 0.90 P2RX7 (0.47) NPC1RAB9AMAPTTP53LMNA
SCHEMBL2760640 0.90 P2RX7 (0.47) NPC1RAB9AMAPTTP53LMNA
SCHEMBL2760776 0.89 PSEN1 (0.41) NPC1RAB9AMAPTTP53AKR1C3
SCHEMBL2760777 0.89 PSEN1 (0.41) NPC1RAB9AMAPTTP53AKR1C3
SCHEMBL2760578 0.85 PSEN1 (0.40) NPC1RAB9AMAPTTP53PSEN1
SCHEMBL2760579 0.85 PSEN1 (0.40) NPC1RAB9AMAPTTP53PSEN1
SCHEMBL2760782 0.84 NPC1 (0.49) NPC1RAB9AMAPTTP53AKR1C3
SCHEMBL2760721 0.80 P2RX3 (0.49) NPC1RAB9AMAPTTP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262766-A2 AMIDE COMPOUNDS, COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2010-12-22 EP disclosed
WO-2009110985-A2 AMIDE COMPOUNDS, COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2009-09-11 WO disclosed