SCHEMBL27611549

SCHEMBL27611549

CC(c1cccc(N)c1)C(C)(C)OC(N)=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CPN1 P15169 1/20 0.41
CPB2 Q96IY4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.38
ADRB2 P07550 5/20 0.38
ADRB3 P13945 3/20 0.38
ADRB1 P08588 2/20 0.38
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
MAPKAPK2 P49137 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
HPGDS O60760 1/20 0.33
PBRM1 Q86U86 1/20 0.33
DDX3X O00571 1/20 0.33
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27389052 0.82 CYP1A2 (0.43) L3MBTL1ALOX5
SCHEMBL28025968 0.79 MEN1 (0.48) L3MBTL1ALDH1A1ALOX5
SCHEMBL8953959 0.78 CYP3A4 (0.37) CPN1CPB2ADRB2ADRB3ADRB1
SCHEMBL1067891 0.76 CPN1 (0.47) CPN1CPB2ADRB2ADRB3ADRB1
SCHEMBL28140608 0.75 CYP17A1 (0.40) L3MBTL1ALDH1A1
SCHEMBL27493803 0.74 ESR1 (0.41) ALDH1A1CA1CA2CA9
SCHEMBL5796124 0.74 APP (0.47) CPN1CPB2ADRB2ADRB3ADRB1
SCHEMBL27647919 0.73 ALOX5 (0.46) ALDH1A1ALOX5
SCHEMBL27510737 0.73 ACACB (0.36) ALOX5
SCHEMBL7336123 0.72 CPN1 (0.43) CPN1CPB2ADRB2ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100348196-C Benzotriaza * as gastrin and cholecystokinin receptor ligands BLACK JAMES FOUNDATION (GB) 2007-11-14 CN disclosed
CN-1585643-A Benzotriazepines as gastrin and cholecystokinin receptor ligands BLACK JAMES FOUNDATION (GB) 2005-02-23 CN disclosed