SCHEMBL27612010

SCHEMBL27612010

C1=Cc2ccc3c4c(ccc3c2CC1)CCCC4

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES1 P23141 4/20 0.40
KIF11 P52732 1/20 0.36
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
BCL2L1 Q07817 1/20 0.32
BAD Q92934 1/20 0.32
GNG2 P59768 1/20 0.32
GNB1 P62873 1/20 0.32
NQO1 P15559 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
STAT3 P40763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27781003 0.84
SCHEMBL28024035 0.79 CES1 (0.37) CES1KIF11GRIA1GRIA2GRIA3
SCHEMBL27697057 0.79
SCHEMBL27994256 0.79
SCHEMBL27855741 0.77 KIF11 (0.33) CES1KIF11BCL2L1BADSTAT3
SCHEMBL27838062 0.77 CES1 (0.31) CES1KIF11STAT3
SCHEMBL27883165 0.74 KIF11 (0.31) CES1KIF11GNG2GNB1
SCHEMBL27837968 0.74 KDM4E (0.31)
SCHEMBL28751592 0.74 HPRT1 (0.37) KIF11BCL2L1BADNQO1
SCHEMBL8666055 0.73 ALDH1A1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103889224-B ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC医疗公司 2017-05-24 CN claimed
CN-107925004-A Organic molecule for organic electro-optic device 西诺拉股份有限公司 2018-04-17 CN disclosed
CN-103450218-B As the indoles three also ring derivatives of CRTH2 receptor antagonist SHANDONG HENRY MEDICAL SCIENCE AND TECHNOLOGY CO., LTD. (CN) 2015-12-23 CN disclosed
CN-102791689-B 3- (heteroaryl-amino) -1,2,3, 4-tetrahydro-9H-carbazole derivatives and their use as prostaglandin D2 receptor modulators ACTELION PHARMACEUTICALS LTD. (CH) 2014-10-29 CN disclosed
CN-101687799-B Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals GRUENENTHAL GMBH 2014-07-23 CN disclosed
CN-103450218-A Indole tricyclic derivative as CRTH2 receptor antagonist SHANDONG HENGLI MEDICAL TECHNOLOGY CO LTD 2013-12-18 CN disclosed
CN-102791689-A 3- (heteroaryl-amino) -1,2,3, 4-tetrahydro-9H-carbazole derivatives and their use as prostaglandin D2 receptor modulators ACTELION PHARMACEUTICALS LTD 2012-11-21 CN disclosed
CN-101687799-A Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals GRUENENTHAL GMBH 2010-03-31 CN disclosed
CN-100500654-C Tetrahydrocarbazole derivatives as ligands for G-protein coupled receptors (GPCRs) ZENTARIS AG (DE) 2009-06-17 CN disclosed
CN-101120002-A Cycloalkyl-fused indole, benzothiophene, benzofuran and indene derivatives WYETH CORP (US) 2008-02-06 CN disclosed
CN-1599720-A Tetrahydrocarbazole derivatives as ligands for G-protein coupled receptors (GPCRs) ZENTARIS AG (DE) 2005-03-23 CN disclosed