SCHEMBL28024035

SCHEMBL28024035

C1=Cc2c(ccc3c4c(ccc23)CCCC4)CC1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.37
KIF11 P52732 1/20 0.36
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
BCL2L1 Q07817 1/20 0.32
BAD Q92934 1/20 0.32
GNG2 P59768 1/20 0.32
GNB1 P62873 1/20 0.32
NQO1 P15559 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
STAT3 P40763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28823601 0.84
SCHEMBL27612010 0.79 CES1 (0.40) CES1KIF11GRIA1GRIA2GRIA3
SCHEMBL27697057 0.79
SCHEMBL27883165 0.78 KIF11 (0.31) CES1KIF11GNG2GNB1
SCHEMBL28022479 0.77 CYP2A6 (0.34)
SCHEMBL27939600 0.76
SCHEMBL8661024 0.73 ALDH1A1 (0.31)
SCHEMBL8691558 0.71 PNMT (0.40)
SCHEMBL28751592 0.70 HPRT1 (0.37) KIF11BCL2L1BADNQO1
SCHEMBL3414799 0.70 HPRT1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903323-A Substituted spiropyrido [1,2-a ] pyrazine derivative and medical application thereof as HIV integrase inhibitor JAPAN TOBACCO INC 2015-09-09 CN disclosed