Pyrrole

Pyrrole

SCHEMBL27612136

c1cc[nH]c1.c1ccc2cc3c(ccc4[nH]ncc43)cc2c1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.42
HSP90AA1 P07900 1/20 0.42
CDK2 P24941 1/20 0.42
HCAR2 Q8TDS4 1/20 0.39
METAP2 P50579 2/20 0.38
FGFR1 P11362 1/20 0.38
DYRK3 O43781 1/20 0.38
CLK1 P49759 1/20 0.38
CLK2 P49760 1/20 0.38
CLK3 P49761 1/20 0.38
GSK3B P49841 1/20 0.38
CDK5 Q00535 1/20 0.38
DYRK1A Q13627 1/20 0.38
CDK5R1 Q15078 1/20 0.38
DYRK2 Q92630 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
NOS1 P29475 3/20 0.38
TRPA1 O75762 2/20 0.38
ALDH1A1 P00352 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30486 0.92 IDO1 (0.48) IDO1HSP90AA1CDK2HCAR2METAP2
Hydrochloric Acid SCHEMBL999376 0.90 IDO1 (0.47) IDO1HSP90AA1CDK2HCAR2METAP2
SCHEMBL4141797 0.77 RAF1 (0.40) IDO1HSP90AA1CDK2MKNK1
SCHEMBL17255318 0.76 HASPIN (0.45) FGFR1CLK1DYRK1A
SCHEMBL29563426 0.76 IDO1 (0.54) IDO1HSP90AA1CDK2METAP2FGFR1
SCHEMBL276443 0.76 IDO1 (0.54) IDO1HSP90AA1CDK2METAP2FGFR1
SCHEMBL29450787 0.73 HPRT1 (0.54) IDO1HSP90AA1CDK2HCAR2METAP2
SCHEMBL27074503 0.73 HPRT1 (0.54) IDO1HSP90AA1CDK2HCAR2METAP2
SCHEMBL7208201 0.73 PTPRC (0.41) IDO1ALDH1A1TDP1
Indazole SCHEMBL15577295 0.72 HSP90AA1 (0.79) IDO1HSP90AA1CDK2METAP2FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976936-A Tetrahydroquinolines MERCK PATENT GMBH (DE) 2007-06-06 CN disclosed
CN-1878556-A Combinations of drugs for the treatment of neoplasms COMBINATORX INC (US) 2006-12-13 CN disclosed
CN-1829509-A Pharmaceutical composition for treating tumors COMBINATORX INC (US) 2006-09-06 CN disclosed
CN-1681511-A Combinations of drugs for the treatment of neoplasms COMBINATORX INC (US) 2005-10-12 CN disclosed