SCHEMBL27615365

SCHEMBL27615365

Cc1cccc2nc(C#N)[nH]c12

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 2/20 0.40
PARP1 P09874 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TSHR P16473 1/20 0.35
AHR P35869 1/20 0.35
AR P10275 1/20 0.35
KIF11 P52732 1/20 0.34
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
DAO P14920 1/20 0.33
DDO Q99489 1/20 0.33
USP8 P40818 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL251068 0.80 PSMB8 (0.41) PSMB8ALDH1A1HTTGAA
SCHEMBL11854195 0.77 PARP1 (0.44) PARP1ALDH1A1TSHRPDE3BPDE3A
SCHEMBL353892 0.75 PARP1 (0.56) PARP1NPC1ALDH1A1HPGDHTT
SCHEMBL31033488 0.75 PARP1 (0.56) PARP1NPC1ALDH1A1HPGDHTT
SCHEMBL24553999 0.75 EGFR (0.39) PARP1NPC1ALDH1A1HPGDHTT
SCHEMBL29733018 0.75 EGFR (0.39) PARP1NPC1ALDH1A1HPGDHTT
SCHEMBL29893903 0.73 KEAP1 (0.42) PSMB8ALDH1A1HPGDRAB9A
SCHEMBL14091258 0.73 GRM5 (0.45) PARP1NPC1ALDH1A1HPGDHTT
Bromide SCHEMBL5318093 0.73 PARP1 (0.55) PARP1NPC1ALDH1A1HPGDHTT
SCHEMBL10960503 0.72 ALDH1A1 (0.48) PSMB8NPC1ALDH1A1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108383880-A Target cumarin-platinum (II) complex and its synthetic method and the application of ovarian cancer drug-resistant strain 玉林师范学院 2018-08-10 CN disclosed
CN-102592040-B The method of drug discovery 基德姆生物科学有限公司 2016-12-21 CN disclosed
CN-102592040-A Drug discovery method KEDDEM BIO SCIENCE LTD 2012-07-18 CN disclosed
CN-1668918-A Methods of Drug Discovery KEDDEM BIO SCIENCE LTD (IL) 2005-09-14 CN disclosed