SCHEMBL27618166

SCHEMBL27618166

COC(=O)c1cc(C(Br)C=O)ccc1OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 2/20 0.48
POLB P06746 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
F2 P00734 1/20 0.48
F7 P08709 1/20 0.48
FOLH1 Q04609 1/20 0.46
HPGD P15428 4/20 0.44
HTT P42858 1/20 0.44
LMNA P02545 2/20 0.44
LRRK2 Q5S007 2/20 0.43
SMPD1 P17405 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
USP2 O75604 1/20 0.43
CTSV O60911 1/20 0.42
CTSL P07711 1/20 0.42
CYP1A2 P05177 1/20 0.42
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27820730 0.88 F2 (0.53) ALDH1A1KDM4EPOLBL3MBTL1F2
SCHEMBL5552677 0.85 F2 (0.51) ALDH1A1KDM4EPOLBL3MBTL1F2
SCHEMBL965193 0.82 F2 (0.49) ALDH1A1KDM4EPOLBL3MBTL1F2
SCHEMBL965192 0.82 F2 (0.49) ALDH1A1KDM4EPOLBL3MBTL1F2
SCHEMBL6874912 0.82 HPGD (0.51) ALDH1A1KDM4EPOLBF2F7
SCHEMBL10477773 0.81 L3MBTL1 (0.43) ALDH1A1KDM4EPOLBL3MBTL1F2
SCHEMBL852240 0.80 ALDH1A1 (0.59) ALDH1A1KDM4EPOLBL3MBTL1FOLH1
SCHEMBL5702073 0.80 FFAR4 (0.50) ALDH1A1KDM4EPOLBL3MBTL1FOLH1
SCHEMBL4416634 0.80 FOLH1 (0.58) ALDH1A1KDM4EPOLBL3MBTL1FOLH1
SCHEMBL5431545 0.79 LRRK2 (0.63) ALDH1A1KDM4EPOLBL3MBTL1FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101239969-B Biphenyl derivatives THERAVANCE INC 2011-07-20 CN disclosed
CN-101239968-B Biphenyl derivatives THERAVANCE INC 2011-07-20 CN disclosed
CN-101239970-B Biphenyl derivatives THERAVANCE INC 2011-07-20 CN disclosed
CN-101239971-B Biphenyl derivatives THERAVANCE INC 2011-07-20 CN disclosed
CN-101239968-A Biphenyl derivatives THERAVANCE INC (US) 2008-08-13 CN disclosed
CN-101239969-A Biphenyl derivatives THERAVANCE INC (US) 2008-08-13 CN disclosed
CN-101239971-A Biphenyl derivatives THERAVANCE INC (US) 2008-08-13 CN disclosed
CN-101239970-A Biphenyl derivatives THERAVANCE INC (US) 2008-08-13 CN disclosed
CN-100378092-C Biphenyl derivatives THERAVANCE INC (US) 2008-04-02 CN disclosed
CN-1759108-A Biphenyl derivatives THERAVANCE INC (US) 2006-04-12 CN disclosed