SCHEMBL27622980

SCHEMBL27622980

CCc1cc(C(=O)O)c([N+](=O)[O-])c(N)c1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
POLB P06746 1/20 0.46
PKM P14618 1/20 0.44
ALDH1A1 P00352 3/20 0.41
GABRP O00591 2/20 0.41
GABRD O14764 2/20 0.41
GABRA1 P14867 2/20 0.41
GABRB1 P18505 2/20 0.41
GABRG2 P18507 2/20 0.41
GABRB3 P28472 2/20 0.41
GABRA5 P31644 2/20 0.41
GABRA3 P34903 2/20 0.41
GABRA2 P47869 2/20 0.41
GABRB2 P47870 2/20 0.41
GABRA4 P48169 2/20 0.41
GABRE P78334 2/20 0.41
GABRA6 Q16445 2/20 0.41
GABRG1 Q8N1C3 2/20 0.41
GABRG3 Q99928 2/20 0.41
GABRQ Q9UN88 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26672390 0.81 HTT (0.41) HTTPOLBPKMALDH1A1GABRP
SCHEMBL8403333 0.81 ALDH1A1 (0.45) HTTPOLBPKMALDH1A1GABRP
SCHEMBL10661895 0.77 ALDH1A1 (0.47) HTTPKMALDH1A1CYP3A4GRIN2D
SCHEMBL10416134 0.76 PKM (0.40) HTTPOLBPKMALDH1A1GABRP
SCHEMBL29141466 0.76 PKM (0.43) HTTPKMALDH1A1TP53CYP1A2
SCHEMBL5161255 0.74 HTT (0.69) HTTPOLBALDH1A1GABRPGABRD
SCHEMBL26963219 0.73 ALDH1A1 (0.55) POLBPKMALDH1A1CYP3A4ALOX15
SCHEMBL30626464 0.73 ALDH1A1 (0.55) POLBPKMALDH1A1CYP3A4ALOX15
SCHEMBL1202500 0.73 PKM (0.47) HTTPKMALDH1A1CYP3A4GRIN2D
SCHEMBL27267409 0.73 HCAR3 (0.43) HTTPKMALDH1A1CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1902159-B Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents AUCKLAND UNISERVICES LTD 2010-06-09 CN disclosed
CN-100546976-C Alkylating agent and they purposes based on N-methyl-p-nitroaniline as prodrug AUCKLAND UNISERVICES LTD (NZ) 2009-10-07 CN disclosed
CN-1902159-A Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents AUCKLAND UNISERVICES LTD (NZ) 2007-01-24 CN disclosed
CN-1711236-A Nitroaniline-based alkylating agents and their use as prodrugs AUCKLAND UNISERVICES LTD (NZ) 2005-12-21 CN disclosed