SCHEMBL27623980

SCHEMBL27623980

O=C(c1ccc(-c2ccccc2)s1)c1ccc(-c2ccccc2)s1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.71
MEN1 O00255 1/20 0.71
POLB P06746 1/20 0.71
KMT2A Q03164 1/20 0.71
HDAC1 Q13547 1/20 0.69
NPC1 O15118 2/20 0.65
KDM4E B2RXH2 1/20 0.65
ALDH1A1 P00352 1/20 0.65
HPGD P15428 1/20 0.65
HDAC6 Q9UBN7 1/20 0.65
PPARG P37231 1/20 0.62
NCOA2 Q15596 1/20 0.62
NCOA1 Q15788 1/20 0.62
NCOA3 Q9Y6Q9 1/20 0.62
ERCC5 P28715 1/20 0.61
FEN1 P39748 1/20 0.61
HSD17B1 P14061 6/20 0.59
HSD17B2 P37059 6/20 0.59
HPGDS O60760 2/20 0.58
HSD11B1 P28845 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12494820 0.90 HSD17B1 (0.66) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL1761545 0.87 RAB9A (0.92) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL10275320 0.85 RAB9A (0.69) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL11913196 0.84 HSD17B1 (0.81) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL11913209 0.84 HSD17B1 (0.57) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL3097763 0.83 RAB9A (0.67) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL2690201 0.83 IKBKB (0.68) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL4128733 0.83 RAB9A (0.67) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL2491267 0.83 RAB9A (1.00) RAB9AMEN1POLBKMT2AHDAC1
SCHEMBL11913205 0.82 HSD17B1 (0.57) RAB9AMEN1POLBKMT2AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN claimed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN claimed
CN-104109155-A Novel compounds TANABE SEIYAKU CO 2014-10-22 CN disclosed
CN-103819465-A Novel compound MITSUBISHI TANABE PHARMA CORP 2014-05-28 CN disclosed
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN disclosed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN disclosed