SCHEMBL27627752

SCHEMBL27627752

CC(=O)Oc1c(-c2ccc(F)cc2)c(-c2ccncc2)c2n1CCC2C

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 13/20 0.45
MAPK11 Q15759 3/20 0.43
KCNH2 Q12809 1/20 0.43
HTR3A P46098 1/20 0.38
MAPK13 O15264 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPK12 P53778 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6218210 0.80 HTR3A (0.57) MAPK14MAPK11KCNH2HTR3AMAPK13
SCHEMBL27627894 0.72 MAPK14 (0.44) MAPK14MAPK11KCNH2HTR3AMAPK13
SCHEMBL27608556 0.72 MAPK14 (0.52) MAPK14MAPK11HTR3AMAPK13CYP2C9
SCHEMBL27627887 0.72 MAPK14 (0.44) MAPK14MAPK11KCNH2HTR3AMAPK13
SCHEMBL27608554 0.71 MAPK14 (0.46) MAPK14MAPK11KCNH2HTR3AMAPK13
SCHEMBL27627904 0.70 HTR3A (0.68) MAPK14MAPK11KCNH2HTR3AMAPK13
SCHEMBL27909189 0.68 KCNK3 (0.37) MAPK14MAPK11KCNH2HTR3A
SCHEMBL27627754 0.65 MAPK14 (0.45) MAPK14MAPK11KCNH2MAPK13MAPK12
SCHEMBL27627755 0.65 MAPK14 (0.45) MAPK14MAPK11KCNH2MAPK13MAPK12
SCHEMBL27627770 0.65 MAPK14 (0.44) MAPK14MAPK11KCNH2MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1701069-A 3,4-disubstituted pyrroles and their for use in treating inflammatory diseases JANSSEN PHARMACEUTICA NV (BE) 2005-11-23 CN disclosed