SCHEMBL27630643

SCHEMBL27630643

CC(NC(=O)OC(C)(C)C)C(=O)NC(C)C(=O)NC(CC(N)=O)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 2/20 0.49
REN P00797 1/20 0.46
BACE1 P56817 6/20 0.46
KMT2A Q03164 2/20 0.44
APP P05067 1/20 0.43
CTSS P25774 3/20 0.42
CTSK P43235 3/20 0.42
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
ATM Q13315 1/20 0.41
GLS O94925 1/20 0.40
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27630641 1.00 ECE1 (0.49) ECE1RENBACE1KMT2AAPP
SCHEMBL19384891 0.96 REN (0.49) ECE1RENBACE1KMT2AAPP
SCHEMBL20677180 0.96 REN (0.49) ECE1RENBACE1KMT2AAPP
SCHEMBL20677179 0.96 REN (0.49) ECE1RENBACE1KMT2AAPP
SCHEMBL3493240 0.90 BACE1 (0.52) RENBACE1APPCTSSCTSK
SCHEMBL30186037 0.89 KMT2A (0.46) RENKMT2ACTSSCTSKCTSL
SCHEMBL29918245 0.87 REN (0.44) RENBACE1KMT2ACTSSCTSK
SCHEMBL29274070 0.87 KMT2A (0.47) RENKMT2ACTSSCTSKCTSL
SCHEMBL29274069 0.87 KMT2A (0.47) RENKMT2ACTSSCTSKCTSL
SCHEMBL999894 0.87 APP (0.49) ECE1APPCTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100381459-C Adriamycin derivative and its preparing method and use CHENGDU NANSHAN PHARMACEUTICAL (CN) 2008-04-16 CN disclosed
CN-1781932-A Adriamycin derivative and its preparing method and use NANSHAN PHARMACEUTICAL CO LTD (CN) 2006-06-07 CN disclosed