SCHEMBL27633488

SCHEMBL27633488

O=C(c1ccn(Cc2cccnc2)c1-c1ccccc1)c1ccn(Cc2cccnc2)c1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHPS P49366 1/20 0.50
ALDH1A1 P00352 4/20 0.48
ADRA1D P25100 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
KDM4E B2RXH2 2/20 0.45
LMNA P02545 2/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
NAPRT Q6XQN6 1/20 0.44
CYP2E1 P05181 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2A6 P11509 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
CYP2C19 P33261 1/20 0.44
P2RX7 Q99572 1/20 0.44
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
NOTUM Q6P988 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3496060 0.77 NOTUM (0.64) ALDH1A1ADRA1DL3MBTL1KDM4ELMNA
SCHEMBL5762448 0.75 THRB (0.51) ALDH1A1KDM4ELMNA
SCHEMBL4273292 0.71 NOTUM (0.52) KDM4EKMT2ANOTUM
SCHEMBL20893846 0.71 TSHR (0.51) DHPSALDH1A1ADRA1DKDM4ENAPRT
SCHEMBL12120857 0.70 HDAC3 (0.57) DHPSKDM4ELMNAHTTNAPRT
SCHEMBL3495559 0.69 CYP19A1 (0.55) ALDH1A1KDM4ELMNANOTUMTSHR
SCHEMBL16220643 0.68 CHRNB2 (0.51) DHPSL3MBTL1KDM4ELMNAMAPK1
SCHEMBL27638474 0.68 ADRA1D (0.43) DHPSALDH1A1ADRA1DL3MBTL1KDM4E
SCHEMBL7809472 0.67 KMT2A (0.60) KDM4EKMT2AHDAC1HDAC2HDAC10
SCHEMBL6840334 0.67 PLAU (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100427472-C Aryl-heteroaromatic compounds, compositions containing them and their use AVENTIS PHARMA SA (FR) 2008-10-22 CN disclosed
CN-1829697-A Aryl-heteroaromatic products, compositions containing same and use thereof AVENTIS PHARMA SA (FR) 2006-09-06 CN disclosed