SCHEMBL27634896

SCHEMBL27634896

N#CCc1nc(-c2ccc(Cl)cc2)cnc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.43
ATR Q13535 1/20 0.42
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
PARP1 P09874 1/20 0.39
CTRC Q99895 3/20 0.39
KMT2A Q03164 4/20 0.38
MAPT P10636 1/20 0.38
MEN1 O00255 3/20 0.37
CA12 O43570 1/20 0.37
ALPL P05186 1/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KDM4E B2RXH2 4/20 0.36
XDH P47989 1/20 0.36
AKR1B1 P15121 1/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
RUNX1 Q01196 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27634968 0.83 KMO (0.47) KMOATRNPC1RAB9ASMN1; SMN2
SCHEMBL4680329 0.80 CDH1 (0.43) KMONPC1CTRCKDM4EALDH1A1
SCHEMBL27655897 0.79 KMO (0.43) KMOATRNPC1RAB9ASMN1; SMN2
SCHEMBL11216316 0.78 ATR (0.53) KMOATRNPC1RAB9ASMN1; SMN2
SCHEMBL27634863 0.77 SMN1; SMN2 (0.47) KMOATRNPC1RAB9ASMN1; SMN2
SCHEMBL27655888 0.75 HPGD (0.47) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL27656038 0.74 ATR (0.41) KMOATRNPC1RAB9ASMN1; SMN2
SCHEMBL27634965 0.74 KMO (0.39) KMOATRNPC1RAB9ASMN1; SMN2
SCHEMBL27655941 0.73 KMT2A (0.46) NPC1RAB9APARP1KMT2AMEN1
SCHEMBL27655896 0.73 ALDH1A1 (0.40) KMOATRNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1809554-A 3-substituted 5,6-diaryl-pyrazine-2-carboxamide and -2-sulfonamide derivatives as cb1 modulators ASTRAZENECA AB (SE) 2006-07-26 CN disclosed