SCHEMBL27636201

SCHEMBL27636201

CC(=O)OC(C)(C)Cn1ccc2c(O)cccc21

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.48
NR3C1 P04150 7/20 0.39
PGR P06401 6/20 0.39
NR3C2 P08235 6/20 0.39
KDM4E B2RXH2 3/20 0.39
HSD17B10 Q99714 1/20 0.39
HTR6 P50406 1/20 0.36
AR P10275 2/20 0.33
GLA P06280 2/20 0.33
LMNA P02545 1/20 0.33
NOTUM Q6P988 1/20 0.33
CYP3A4 P08684 1/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5015442 0.77 HTR2C (0.49) HTR2CKDM4EHSD17B10HTR6ALDH1A1
SCHEMBL27656185 0.76 NR3C1 (0.33) NR3C1KDM4EHSD17B10
SCHEMBL28760998 0.75 HTR2C (0.57) HTR2CHTR6THRBALDH1A1
SCHEMBL27657110 0.73 MTNR1A (0.39) KDM4EHSD17B10ARALDH1A1
SCHEMBL4323537 0.71 HTR2C (0.63) HTR2CNR3C1PGRNR3C2KDM4E
SCHEMBL29751560 0.71 HTR2C (0.63) HTR2CNR3C1PGRNR3C2KDM4E
SCHEMBL3169119 0.70 KMT2A (0.57) HTR2CKDM4EHTR6GLAALDH1A1
SCHEMBL3874161 0.69 ALDH1A1 (0.53) HTR2CKDM4ELMNACYP3A4ALDH1A1
SCHEMBL6385676 0.69 HTR2C (0.57) HTR2CKDM4ELMNAALDH1A1
SCHEMBL4321418 0.69 HTR2C (0.60) HTR2CKDM4EHSD17B10HTR6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1816550-B Indolyl derivatives substituted with a thiazole ring and their use as PPAR modulators HOFFMANN LA ROCHE 2010-04-28 CN disclosed
CN-1816550-A Indolyl derivatives substituted with a thiazole ring and their use as ppar modulators HOFFMANN LA ROCHE (CH) 2006-08-09 CN disclosed