SCHEMBL27636205

SCHEMBL27636205

N#CCCNc1cc[nH]c1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.47
HTT P42858 1/20 0.47
ALDH1A1 P00352 1/20 0.47
THRB P10828 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11252528 0.77 GAA (0.70) GAAHTTALDH1A1THRB
SCHEMBL27878117 0.74
SCHEMBL141474 0.71 GAA (0.58) GAAHTTALDH1A1THRB
SCHEMBL6554127 0.71 GAA (0.58) GAAHTTALDH1A1THRB
SCHEMBL27515091 0.71 CYP1A2 (0.40) ALDH1A1
SCHEMBL11252585 0.69 HTT (0.61) GAAHTTALDH1A1THRB
SCHEMBL5028293 0.69 GAA (0.61) GAAHTTALDH1A1THRB
SCHEMBL4615070 0.69 ADRA2A (0.41) GAAALDH1A1
SCHEMBL28189161 0.69
SCHEMBL6161907 0.68 THRB (0.66) GAAHTTALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1832925-B New P2X7 receptor avtagonists and their use ASTRAZENECA AB 2010-05-05 CN disclosed
CN-101111488-A Novel compounds ASTRAZENECA AB (SE) 2008-01-23 CN disclosed
CN-1832925-A New p2x7 receptor avtagonists and their use ASTRAZENECA AB (SE) 2006-09-13 CN disclosed