SCHEMBL276364

SCHEMBL276364

[CH]1CNCCN1Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.56
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
HIF1A Q16665 1/20 0.44
PIM1 P11309 1/20 0.40
SLC6A4 P31645 4/20 0.40
SLC6A2 P23975 3/20 0.40
HTR3A P46098 2/20 0.40
CXCR4 P61073 1/20 0.40
CYP2D6 P10635 1/20 0.40
MC4R P32245 1/20 0.39
GAA P10253 1/20 0.39
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
ADRB1 P08588 1/20 0.38
HTR3D Q70Z44 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16598868 0.82 ALDH1A1 (0.47) SIGMAR1MEN1ALDH1A1CYP2C9KMT2A
SCHEMBL16598932 0.78 SIGMAR1 (0.51) SIGMAR1KMT2ACYP2D6ADRB1
SCHEMBL16598812 0.78 HPGD (0.40) SIGMAR1MEN1ALDH1A1KMT2AHTR3A
SCHEMBL2228270 0.76 SIGMAR1 (0.56) SIGMAR1ALDH1A1MC4RDRD4
SCHEMBL16599267 0.75 DBH (0.36) ALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL16598887 0.75 TACR1 (0.35) SIGMAR1MEN1KMT2ACXCR4ADRB1
SCHEMBL4903098 0.75 ALDH1A1 (0.46) SIGMAR1MEN1ALDH1A1TSHRCYP2C19
SCHEMBL4906727 0.73 MAPT (0.40) MEN1ALDH1A1CYP2C9TSHRCYP2C19
SCHEMBL6138636 0.72 SIGMAR1 (1.00) SIGMAR1MEN1ALDH1A1CYP2C9TSHR
SCHEMBL152631 0.72 SIGMAR1 (1.00) SIGMAR1MEN1ALDH1A1CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 259 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118125997-A Pterocarpus stilbene paeonol chalcone amide derivative, preparation method and medical application thereof 安徽中医药大学 2024-06-04 CN claimed
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN claimed
CN-116102565-A Isolamine-containing spirochromone compound and preparation method and application thereof 贵州大学 2023-05-12 CN claimed
CN-113717201-B (+/-) -Marinopyrole A derivative and preparation method and application thereof 植恩生物技术股份有限公司 2022-12-16 CN claimed
CN-115260046-A Abietate compound and preparation method and application thereof 贵州大学 2022-11-01 CN claimed
CN-115141208-A Podophyllotoxin compound containing various ester group structures and preparation method and application thereof 贵州大学 2022-10-04 CN claimed
CN-114920722-A 7-hydroxy-3-acetyl coumarin oxime compound, preparation method and medical application thereof 何黎琴 2022-08-19 CN claimed
CN-113717201-A (+/-) -Marinopyrole A derivative and preparation method and application thereof 植恩生物技术股份有限公司 2021-11-30 CN claimed
CN-112707843-A Novel paeonol oxime compound, preparation method and medical application thereof 何黎琴 2021-04-27 CN claimed
CN-112624931-A Pterostilbene amine compounds containing isopropanol aromatic ether structure and preparation method and application thereof 贵州大学 2021-04-09 CN claimed
EP-0567982-B1 Azole compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-07-01 EP claimed
EP-0804428-A1 BIS-SULFONAMIDE HYDROXYETHYLAMINO RETROVIRAL PROTEASE INHIBITORS G.D. SEARLE & CO. (US) 1997-11-05 EP claimed
EP-0347678-B1 1,4-Dihydropyridine threonin derivatives and process for their preparation BAYER AG (DE) 1997-02-26 EP claimed
US-5604294-A IMMUNOSUPRESSIVE, ANTIMICROBIAL, ANTIFUNGAL, ANTIVIRAL, ANTI-INFLAMMATORY AND ANTIPROLIFERATIVE ACTIVITY ABBOTT LABORATORIES 1997-02-18 US claimed
WO-1996022287-A1 BIS-SULFONAMIDE HYDROXYETHYLAMINO RETROVIRAL PROTEASE INHIBITORS G.D. SEARLE & CO. (US) 1996-07-25 WO claimed
WO-1994021635-A1 MACROCYCLIC IMMUNOMODULATORS ABBOTT LABORATORIES (US) 1994-09-29 WO claimed
US-4939142-A Substituted styrene derivatives EGIS GYOGYSZERGYAR (HU) 1990-07-03 US claimed
EP-0347678-A2 1,4-Dihydropyridine threonin derivatives and process for their preparation BAYER AG (DE) 1989-12-27 EP claimed
US-4786638-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS AMERICAN HOME PRODUCTS CORPORATION (US) 1988-11-22 US claimed
US-4395413-A NICOTINE ANTIALLERGEN, ANESTHETIC, ANALGESIC, HYPOTENSIVE, AND ANTIULCER AGENT EGYT GYOGYSZERVEGYESZETI GYAR (HU) 1983-07-26 US claimed