SCHEMBL6138636

SCHEMBL6138636

c1ccc(CN2CCNCC2)cc1.c1ccc(CN2CCNCC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 1.00
MEN1 O00255 2/20 0.68
KMT2A Q03164 2/20 0.68
ALDH1A1 P00352 1/20 0.68
CYP2C9 P11712 1/20 0.68
TSHR P16473 1/20 0.68
CYP2C19 P33261 1/20 0.68
HIF1A Q16665 1/20 0.68
CXCR4 P61073 9/20 0.64
CHRM2 P08172 1/20 0.63
CHRM1 P11229 1/20 0.63
ADRA2C P18825 1/20 0.63
CCR2 P41597 1/20 0.63
CXCL12 P48061 1/20 0.63
BLM P54132 1/20 0.63
TDP1 Q9NUW8 1/20 0.63
HRH3 Q9Y5N1 1/20 0.63
MC4R P32245 1/20 0.59
DRD4 P21917 1/20 0.57
LMNA P02545 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL83548 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL276363 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
Benzene SCHEMBL27761330 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL152631 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL7062479 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL7573306 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
Hydrochloric Acid SCHEMBL2223234 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL8145866 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL10063607 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
Ammonia Solution, Strong SCHEMBL28172574 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1277746-B1 N-benzylpiperazine derivatives, process for their preparation and pharmaceutical compositions thereof SERVIER LAB (FR) 2005-05-11 EP disclosed
EP-1277746-A3 N-benzylpiperazine derivatives, process for their preparation and pharmaceutical compositions thereof Les Laboratoires Servier (FR) 2003-08-13 EP disclosed
EP-1277746-A2 N-benzylpiperazine derivatives, process for their preparation and pharmaceutical compositions thereof Les Laboratoires Servier (FR) 2003-01-22 EP disclosed