SCHEMBL27636766

SCHEMBL27636766

CC(=O)c1ccc(OS(=O)(=O)C(F)(F)F)cc1CN

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.53
HTR1D P28221 5/20 0.45
HTR1A P08908 4/20 0.45
HTR1B P28222 4/20 0.45
CXCR2 P25025 2/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CXCR1 P25024 1/20 0.39
MAOB P27338 4/20 0.38
MAOA P21397 1/20 0.36
STS P08842 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
DRD2 P14416 2/20 0.36
DRD3 P35462 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19179854 0.84 HSD11B1 (0.56) HSD11B1HTR1DHTR1AHTR1BCXCR2
SCHEMBL1748180 0.81 HSD11B1 (0.56) HSD11B1HTR1DHTR1AHTR1BCXCR2
SCHEMBL3362412 0.79 HSD11B1 (0.55) HSD11B1HTR1DHTR1AHTR1BCXCR2
SCHEMBL27351302 0.78 HSD11B1 (0.56) HSD11B1HTR1DHTR1AHTR1BCXCR2
SCHEMBL18097828 0.78 HSD11B1 (0.56) HSD11B1HTR1DHTR1AHTR1BCXCR2
SCHEMBL3904794 0.75 HSD11B1 (0.43) HSD11B1HTR1DHTR1AHTR1BCXCR2
SCHEMBL5565709 0.73 ALDH1A1 (0.51) HSD11B1HTR1DHTR1AHTR1BCXCR2
SCHEMBL20526582 0.73 HTR1D (0.46) HSD11B1HTR1DHTR1AHTR1BCA1
SCHEMBL6284793 0.72 CXCR2 (0.43) HSD11B1HTR1DHTR1AHTR1BCXCR2
SCHEMBL5569165 0.72 HSD11B1 (0.47) HSD11B1HTR1DCXCR2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1816531-A Process for the preparation of aryl alkyl acid derivatives and their use for the treatment of obesity BAYER PHARMACEUTICALS CORP (US) 2006-08-09 CN disclosed