SCHEMBL27640709

SCHEMBL27640709

Cc1nc(C(F)(F)F)sc1CCl

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 2/20 0.36
PPARA Q07869 2/20 0.36
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25164661 0.82 PPARD (0.37) PPARDPPARA
SCHEMBL15211249 0.80 PPARD (0.39) PPARDPPARA
SCHEMBL25025569 0.77 SRC (0.39) PPARDPPARAMAPT
SCHEMBL4471873 0.73 MAPT (0.45) PPARDPPARAMAPT
SCHEMBL28996471 0.72
SCHEMBL24137968 0.72 PPARD (0.34) PPARDPPARA
SCHEMBL1846903 0.72
SCHEMBL13841474 0.72 NOS1 (0.42)
Hydrochloric Acid SCHEMBL4858282 0.70 ALDH1A1 (0.39)
SCHEMBL977726 0.70 MAPT (0.59) PPARDPPARAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1972916-B Cinnamide compounds EISAI R&D MAN CO LTD 2013-03-27 CN disclosed
CN-101723900-B Cinnamide compounds EISAI R&D MAN CO LTD 2012-08-22 CN disclosed
CN-101830863-B Method and intermediate compound for preparing ligand of PPAR (Peroxisome Proliferator-Activated Receptor) delta SEOUL NAT UNIV IND FOUNDATION 2011-06-22 CN disclosed
CN-101193876-B Process for preparing ligands for PPAR δ and intermediate compounds useful for preparing the ligands SEOUL NAT UNIV IND FOUNDATION 2011-05-11 CN disclosed
CN-101830863-A The method and the intermediate compound that is used to prepare this part of the part of preparation PPAR δ SEOUL NAT UNIV IND FOUNDATION 2010-09-15 CN disclosed
CN-101723900-A Cinnamide compounds EISAI R&D MAN CO LTD 2010-06-09 CN disclosed
CN-100457744-C Process for preparing thiazole derivative and the intermediate compounds for preparing the same SEOUL NAT UNIV IND FOUNDATION (KR) 2009-02-04 CN disclosed
CN-101193876-A Process for preparing ligands for PPAR δ and intermediate compounds useful for preparing the ligands JIANG XIANZHONG (KR) 2008-06-04 CN disclosed
CN-1972916-A Cinnamide compounds EISAI R&D MAN CO LTD (JP) 2007-05-30 CN disclosed
CN-1750820-A Thiazole and oxazole derivatives which modulate PPAR activity WARNER LAMBERT CO (US) 2006-03-22 CN disclosed
CN-1649854-A Process for preparing thiazole derivative and the intermediate compounds for preparing the same HEONJOONG KANG (KR) 2005-08-03 CN disclosed